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1-methyl-8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(1S,2R)-N2-butyl-N1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N1-methylcyclohexane-1,2-dicarboxamide
1-[(2,4-difluorophenyl)methyl]-5-[4-(2-methylphenyl)piperazin-1-yl]azepan-2-one
9-(2-methoxyethyl)-1-methyl-4-(piperidine-1-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(oxolan-2-ylmethyl)acetamide
N-[3-(4-{[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
5-{[(1-hydroxycyclohexyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-(1H-imidazol-4-yl)-2-(1H-pyrrol-1-yl)-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]propan-1-one
4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-N-cycloheptylpiperidine-1-carboxamide
3-fluoro-N,6-dimethyl-N-(quinolin-5-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
2-cyclopropyl-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-3,4-dihydropyrimidin-4-one
2-(4-methoxyphenoxymethyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
(1R,5R)-N,N-dimethyl-6-(5-oxo-5-phenylpentanoyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
2-{[1-(2-methoxyphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
N-cyclopropyl-3-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(2,3-dihydroxypropyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(1H-imidazol-1-yl)propanamide
2-(2-hydroxyethyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
N-[(4-acetylmorpholin-2-yl)methyl]-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
4-[3-(benzyloxy)piperidin-1-yl]-6-ethylpyrimidine
6-fluoro-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]quinolin-4-ol
N-[3-(1H-imidazol-1-yl)propyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-[3-(furan-2-yl)phenyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
N4-[3-(cyclohexylsulfanyl)propyl]-2-methylpyrimidine-4,6-diamine
3-[1-(2-oxo-1,2-dihydroquinoline-4-carbonyl)piperidin-3-yl]benzoic acid
N-cyclohexyl-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1S,5R)-3-(2-phenylethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 4-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]piperidine-1-carboxylate
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
(3R,9aR)-8-(2-fluorobenzenesulfonyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-methyl-4-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
N-(5-carbamoyl-2-methylphenyl)-10-oxo-3,9-diazaspiro[5.6]dodecane-3-carboxamide
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-(thian-4-yl)piperazine
N-benzyl-2-(2-oxopiperidin-1-yl)-N-(2-phenylethyl)acetamide
8-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(2R,3R,6R)-N-butyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-[(2R)-1-hydroxy-1,1-diphenylpropan-2-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N'-(2-fluoro-5-methylphenyl)-N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]butanediamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
9-[(3-methylpyridin-4-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-hydroxyethyl)-N-methyl-1-(1-{[1-(propan-2-yl)-1,2,3,4-tetrahydroquinolin-6-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(methylsulfanyl)propan-1-one
6-ethoxy-3-[(3-hydroxyazetidin-1-yl)methyl]-1,2-dihydroquinolin-2-one