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2-(4-chlorophenoxy)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
2-[(cyclopentylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)-2-(1H-pyrazol-1-yl)benzamide
[(2-butyl-1H-imidazol-4-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
N-ethyl-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxamide
4-methyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidin-2-amine
2-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
2-(morpholin-4-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-(pyridin-3-yl)acetamide
7-{9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3,5-dimethoxy-2-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}benzoic acid
N-(propan-2-yl)-1-{2-[1-(thiophene-2-sulfonyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
N-[(1-hydroxycyclohexyl)methyl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-2H-1,3-benzodioxole-5-carboxamide
2-{1-[(4-fluorophenyl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-5-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
4-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)-1,4-oxazepane
2-[2-({methyl[(2-methylpyridin-4-yl)methyl]amino}methyl)phenyl]-6-(oxolan-2-yl)-3,4-dihydropyrimidin-4-one
N-[2-(4-ethylmorpholin-2-yl)ethyl]-2-(2-methyl-1H-indol-3-yl)acetamide
1-[({[(1R,2S,5R)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl]methyl}carbamoyl)methyl]piperidine-4-carboxamide
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-N-(pyridin-3-ylmethyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-4-methyl-N-[(3S)-2-oxoazepan-3-yl]-1,2,5-oxadiazole-3-carboxamide
1-[2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)ethyl]cyclopentan-1-ol
5-(4,5-dimethylfuran-2-yl)-1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazole
2-amino-4-[2-(ethylamino)pyrimidin-5-yl]-5-propyl-6-(pyridin-3-yl)pyridine-3-carbonitrile
6-{methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-methyl-5-[({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2,4-oxadiazole-3-carboxamide
8-(1H-pyrazole-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-ethyl-2-({4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}methyl)-1,3-thiazole
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-benzyl-N-[(1R,2R)-2-hydroxycyclohexyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-[4-(3-methoxyphenyl)phenyl]piperidin-4-amine
3-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
ethyl 2-({3-[(1H-imidazol-2-ylmethyl)carbamoyl]phenyl}amino)acetate
{5-chloro-7-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
9-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
methyl 2-(4-{imidazo[1,2-a]pyridine-2-carbonyl}-2-oxopiperazin-1-yl)acetate
2-[2-(4-methoxyphenoxymethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-(4-methoxyphenyl)-5-(3-methylthiophene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[1-(2,3-dihydro-1H-inden-4-yl)-5-(1,4-dioxan-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
3-ethyl-1-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-1H-pyrazole-5-carboxamide
3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-4-methylpyridine
(3S,4S)-4-propyl-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidine-3-carboxylic acid
[2-({4-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperazin-1-yl}methyl)phenyl]methanol
2-({[(3R,4R)-1-(2-fluoro-4-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-amino-4-(2-butyl-5-chloro-1H-imidazol-4-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-cyclopropyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
4-methyl-2-{4-[2-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}-6-(propan-2-yl)quinazoline
N4-[2-(pyrrolidine-1-sulfonyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine