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4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(trifluoromethyl)morpholine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(1H-imidazol-1-yl)ethyl]acetamide
2-[8-(2,5-dimethylfuran-3-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
2-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine
2-(2-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)ethan-1-ol
N-{4-[2-(1H-1,2,4-triazol-1-yl)propanamido]phenyl}pentanamide
N-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(pyrimidin-4-ylmethyl)-1H-pyrazole-3-carboxamide
5,8-dimethyl-2-({[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]amino}methyl)quinolin-4-ol
(6R)-6-[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]-1,3-diazinane-2,4-dione
6-{2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}-1H-indazole
1-methyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1H-imidazole-2-carboxamide
1-[3-(4-fluorophenoxy)propyl]-4-(piperidine-3-carbonyl)piperazine
1-(furan-2-carbonyl)-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepane
3-(3-hydroxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]piperidin-4-ol
dimethyl(3-{2-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-7-fluoro-2-methylquinoline-4-carboxamide
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[3-(4-methylphenyl)propanoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1,2-dimethyl-4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-amine
1-(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
2-[1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-(2,5-difluorobenzoyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
methyl 3-(cyclobutylmethoxy)-5-(morpholine-4-carbonyl)benzoate
5-(2,1,3-benzothiadiazol-4-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
1-{[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
methyl 6-{4-[4-(methoxycarbonyl)phenyl]piperazin-1-yl}pyrimidine-4-carboxylate
N-[2-(1-hydroxycyclopentyl)ethyl]-N-methylfuran-3-carboxamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
3-[2-(2,4-difluorophenyl)ethyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(1H-imidazol-1-ylmethyl)piperidine
1,9-dimethyl-4-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-1,4,9-triazaspiro[5.5]undecane
2-(5-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2S,4R)-4-amino-1-[2-(dimethyl-1,3-thiazol-4-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
5-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-2-methylphenol
1-(5-chloropyridin-2-yl)-4-(1H-imidazol-2-ylmethyl)piperazine
2-(1-ethylpiperidin-4-yl)-N-[(4-hydroxyphenyl)methyl]-N-(pyridin-4-ylmethyl)acetamide
1-(3,3-diphenylpiperidin-1-yl)-2-(1H-imidazol-1-yl)ethan-1-one
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
4-{1-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]ethyl}morpholine
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethan-1-one
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyridin-2-ylsulfanyl)acetamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-N-(propan-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
2-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
5,8-dimethyl-2-({[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)quinolin-4-ol