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3-{[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-{1-[(4-methylphenyl)methyl]cyclopropyl}benzamide
1-(furan-2-carbonyl)-4-[4-(1H-imidazol-1-yl)benzoyl]-1,4-diazepane
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-cyclopropylacetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
3-{[5-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methyl-4H-1,2,4-triazole
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)furan-3-carboxamide
N-{2-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
(2S,4R)-N-cycloheptyl-4-(1H-1,2,3,4-tetrazol-1-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
2-[(2-methylprop-2-en-1-yl)oxy]-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]benzamide
N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}thian-4-amine
1-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
N-({1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-3-yl}methyl)-2-(2-methoxyphenoxy)acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(2-fluorophenoxy)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxylic acid
6-[(diethylamino)methyl]-N-(oxan-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-{2-[1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-2-yl]ethyl}phenol
2-({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
dimethyl({5-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]furan-2-yl}methyl)amine
3-[2-(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
2-{2-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
8-(5-chlorothiophene-2-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
6-{[(3-fluorophenyl)methyl]amino}-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
3-[1-(2-fluoro-6-hydroxybenzoyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
2-(4-acetylphenoxy)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
2-[(3-{[2-(pyridin-3-yloxy)propyl]carbamoyl}phenyl)amino]acetic acid
5-[2-(benzenesulfonyl)ethyl]-1-[(4-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazole
N,5-dimethyl-N-(2-phenylethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}butanamide
4-(cyclopropylmethyl)-1-(1-methyl-1H-indole-2-carbonyl)-1,4-diazepan-5-one
6-({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}azetidin-3-ol
(1S,4S)-5-[(2R)-2-amino-3-methylbutanoyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
8-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-N-(1,3-thiazol-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
1-(2-methylpropyl)-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
1-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-(pyridin-3-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-ethyl-4-phenyl-9-propanoyl-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]piperazin-1-yl}-5-ethylpyrimidine
(3S,4R)-1-(3-fluoro-4-methylbenzoyl)-4-methylpiperidine-3,4-diol
1-(carbamoylmethyl)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methylpiperidine-3-carboxamide
6-methyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]quinoline
3,5,7-trimethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-indole-2-carboxamide