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1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(ethylsulfanyl)propan-1-one
4-[4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-ethylpyrimidin-2-yl]morpholine
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
(1R,7S)-N-methyl-4-oxo-3-(pentan-3-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(pyridine-4-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3S,4R)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-ethyl-1H-imidazole
1-propyl-5-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-1,2,4-triazole
3-[5-(2,3-dihydro-1H-inden-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
7-methoxy-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(5-fluoro-2-methoxyphenyl)-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
2-butyl-8-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
4-{[2-(carbamoylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzoic acid
(3S,4S)-1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
(4aR,7aS)-1-acetyl-4-(3-ethyl-1,2-oxazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1'-(2-ethylpyrimidine-5-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-9H-purin-6-amine
1-[(3-fluorophenyl)methyl]-5-(2-methoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
1-[2-(4-chlorophenyl)ethyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
2-[3-(2,5-dimethoxyphenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-(naphthalen-1-yl)-5-[1-(piperidin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]pyrimidine
1-ethyl-N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-ethyl-N2,N2-dimethyl-N4-[1-(morpholin-4-yl)propan-2-yl]pyrimidine-2,4-diamine
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
N-[4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
3-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-(6-methoxy-2H-1,3-benzodioxol-5-yl)urea
N-(4-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}phenyl)acetamide
2-(2-{[2-(dimethylamino)ethyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N3,N3-diethyl-N1-(1-methyl-1H-1,3-benzodiazol-5-yl)piperidine-1,3-dicarboxamide
3-ethyl-5-[(2S)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-4-sulfamoylbenzamide
2-(2-chloro-4-fluorophenoxymethyl)-N-[2-(1H-imidazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylpyridine-4-carboxamide
3-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N-(2-methoxyethyl)-1,3,7-trimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
(1S,5R)-3-(butane-1-sulfonyl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 4-[4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-amido]piperidine-1-carboxylate
1-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
5-(4-methyl-1,4-diazepan-1-yl)-2-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-cyclobutylpiperidine
2-[2-amino-6-(thiophen-2-ylsulfanyl)pyrimidin-4-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(2R)-2-amino-1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}propan-1-one
1-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)methyl]furan-2-carboxamide
5-acetyl-2,4-dimethyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1H-pyrrole-3-carboxamide