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4-phenoxy-1-[2-(1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
4-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
6-{3-[(3aS,6aS)-1-(2-phenylethyl)-octahydropyrrolo[2,3-c]pyrrol-5-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
5-[3,5-bis(trifluoromethyl)benzoyl]-1-(cyclopropylmethyl)-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[2-({2-[5-(2-chlorophenyl)furan-2-yl]-1H-imidazol-1-yl}methyl)morpholin-4-yl]ethan-1-one
1-cyclohexyl-N3-methyl-4-oxo-N5-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
8-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-{4-cyclohexyl-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
7-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2-methoxyethyl)-2-(morpholin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
N-({1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl}methyl)-4-fluorobenzamide
1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}benzenesulfonyl)pyrrolidine
1-(2-methoxybenzoyl)-4-(2,4,5-trimethylbenzoyl)piperazine
(2E)-N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
6-methoxy-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 1-{[(1-methyl-3-phenyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazole-3-carboxylate
[(3R,4R)-1-methanesulfonyl-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(4-chloro-2-fluorobenzoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-3-yl)piperazine
N,N-dimethyl-2-[2-({[(1-methyl-1H-imidazol-2-yl)methyl](propyl)carbamoyl}amino)phenyl]acetamide
3-{[1-(4-hydroxy-1-methylpiperidine-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(thiophen-3-yl)acetamide
8-{2-[(3-hydroxyphenyl)amino]-6-methylpyrimidin-4-yl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(3R,4S)-4-{4-[(6-chloro-2H-chromen-3-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
N-methyl-2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethane-1-sulfonamide
4-[3-(1,3-benzothiazol-2-ylmethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
2-cyclopentyl-N-[2-(dimethylamino)ethyl]-N-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}acetamide
N5-cyclopropyl-N6-(2-methylprop-2-en-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
3-(5-{5-methylimidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-3-yl)pyridazine
3-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)piperidin-2-one
[4-(5-propylpyrimidin-2-yl)phenyl]methanol
9-{[2-(5-methylfuran-2-yl)phenyl]methyl}-3-oxa-9-azaspiro[5.5]undecane
(3S,4R)-1-(2,6-diaminopyrimidin-4-yl)-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2,6-dimethyl-N-(2-methylpropyl)pyrimidine-4-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-methyl-1H-pyrazole-3-carboxamide
1-[1-(5-chloropyridin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-2,5-dimethoxy-N-(pyridin-3-ylmethyl)benzamide
2-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one