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[3-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)phenyl]methanol
5-(4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}phenoxy)-1-azabicyclo[3.2.1]octane
3-[4-({3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)phenyl]prop-2-yn-1-ol
(butan-2-yl)[(3-chlorophenyl)methyl](1H-imidazol-2-ylmethyl)amine
2-{4-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
(3R,4R)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
methyl 3-cyclohexaneamido-6-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
1-[(3-methylpyridin-2-yl)methyl]-4-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperazine
N-[(2-aminopyridin-3-yl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
[(3R,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
7-(3-ethenylphenyl)pyrazolo[1,5-a]pyridine
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
8-acetyl-2-[(3,5-dimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-6-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(4-chloro-3-{[cyclopropyl(pyridin-3-ylmethyl)carbamoyl]amino}phenyl)-2-methoxyacetamide
8-(morpholine-4-sulfonyl)-2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
2-[2-(dimethylamino)ethyl]-8-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
(3S,9aR)-8-[(2-fluoro-5-methylphenyl)methyl]-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-methyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)propanoic acid
4-{4-[(4-methylphenyl)methyl]piperazin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2-(2-methoxyethyl)pyrimidine
2-[(2-fluorophenyl)methyl]-4-[4-(2-phenylpropyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(3S,4R)-3-ethyl-1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-4-methylpiperidin-4-ol
2-[1-cyclopentyl-4-(cyclopropylmethyl)piperazin-2-yl]ethan-1-ol
1-propanoyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N,6-dimethylpyrimidin-4-amine
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[1-(thian-4-yl)piperidin-4-yl]acetamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl][(5-cyclopropyl-1,2-oxazol-3-yl)methyl]methylamine
6-[4-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-2-cyclopropyl-1,3-benzoxazole
(3S,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-chloro-3-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
N-{2-[methyl(phenyl)amino]ethyl}-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
4-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyridine
N-methyl-5-[(methylsulfanyl)methyl]-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}furan-2-carboxamide
ethyl 4-[(3S,4R)-3-acetamido-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]piperidine-1-carboxylate
(2E)-3-(2-chlorophenyl)-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]prop-2-enamide
N-[(3S,4R)-4-propyl-1-[2-(pyridin-4-yl)acetyl]pyrrolidin-3-yl]acetamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]cyclopentanecarboxamide
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-1-ethylpiperidine
2-cyclopropyl-9-(cyclopropylmethyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5,6-dimethylpyrimidine
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}ethan-1-one
1-{1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carbonyl}-1,4-diazepan-5-one
methyl[(3-methylpyridin-4-yl)methyl]{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
2-methoxy-1-[1'-(5-methylpyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-(4-methoxyphenoxymethyl)-1-(1,3-thiazol-4-ylmethyl)piperidine