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4-(1H-1,2,3-benzotriazole-5-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{3-[hydroxy(phenyl)methyl]-5-(1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-(1-benzyl-4-hydroxypiperidin-4-yl)-N-[2-(2-fluorophenyl)ethyl]-1-benzofuran-2-carboxamide
(2R,5R)-1-(dimethyl-1,3-thiazole-4-carbonyl)-2,5-dimethyl-4-(prop-2-en-1-yl)piperazine
5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]-1-oxaspiro[4.5]decan-2-one
4-[(4-chlorophenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-3-ol
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-benzyl-N-cyclopropylpyrrolidine-2-carboxamide
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]furan-2-carboxamide
4-chloro-N-[2-(2-ethoxyphenoxy)ethyl]-N,1-dimethyl-1H-pyrazole-5-carboxamide
N-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-N-methylthian-4-amine
1-methyl-3-({3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)piperidine
N-(2-methylbutyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
(2R,6R)-4-[3-(morpholin-4-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)furan-3-carboxamide
N,N-dimethyl-5-({3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyridin-2-amine
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(piperidin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
1-{[1-(5-chloro-2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-2-one
6-chloro-N-[2-(3-ethoxyphenoxy)ethyl]-N,2-dimethylimidazo[1,2-a]pyridine-3-carboxamide
5-(3-chlorophenyl)-3-[4-(pyridin-2-yl)piperazin-1-yl]-1,2,4-triazine
2-[4-(oxolane-3-carbonyl)piperazin-1-yl]benzonitrile
(3S)-1-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)pyrrolidin-3-ol
1-(2-methoxyphenyl)-4-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}piperazine
(1R,5S)-N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-[(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
1-[3-(1,2-oxazolidin-2-yl)propanoyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
(2R)-2-{[6-(2-chlorophenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
2-{4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]morpholin-3-yl}acetic acid
3-{[1-(5-ethyl-2-methylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}benzoic acid
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
[(2-ethoxyphenyl)methyl](ethyl)[(4-methanesulfonylphenyl)methyl]amine
1-benzyl-5-{[(3-fluoro-4-methylphenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
[1-(2-aminopyridine-4-carbonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
14-(4-methoxy-3-methylphenyl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
8-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
2-{1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
N-(2,5-dimethylphenyl)-N'-[(4-sulfamoylphenyl)methyl]propanediamide
N-(4-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)carbamoyl}phenyl)-2-methylfuran-3-carboxamide
2-{[4-(4-methanesulfonylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
(2H-1,3-benzodioxol-5-ylmethyl)({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}butanamide
methyl 3-{4-[(4-methoxyphenyl)methyl]-3-oxopiperazine-1-carbonyl}benzoate
N-{[(2S,4S)-4-fluoro-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]methyl}methanesulfonamide
5-amino-4-chloro-N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
2,3-dimethyl-6-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]quinoxaline
1-(2-methoxyphenyl)-4-[1-(2-propoxyethyl)piperidin-3-yl]piperazine