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3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-5-propyl-1,2-oxazole
2-[4-(1H-imidazol-2-ylmethyl)piperazin-1-yl]-4-(propan-2-yl)-6-(trifluoromethyl)pyrimidine
{1-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
2-{2-methyl-3-[({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1H-indol-1-yl}acetamide
4-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}piperazin-2-one
N-(2,3-dimethylphenyl)-2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-{2-[5-methyl-4-({methyl[3-(5-methylfuran-2-yl)butyl]amino}methyl)-1,3-oxazol-2-yl]phenyl}methanesulfonamide
8-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
[(3R,4R)-4-[(dimethylamino)methyl]-1-(1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]methanol
4-[(2-fluorophenyl)methyl]-1-[2-(trifluoromethyl)benzoyl]-1,4-diazepan-5-one
2-(3-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-3-yl}phenyl)-1-methyl-1H-imidazole
(2S)-2-[(2,3-dimethylquinoxalin-6-yl)formamido]-3-(pyridin-4-yl)propanoic acid
(1S,5R)-6-(cyclobutylmethyl)-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(dimethylamino)-N-(2-methoxyethyl)-2-(3-methylphenyl)acetamide
2-(3-{4-[1-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}phenoxy)acetamide
3-(4-hydroxyphenyl)-1-[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
1-cyclohexyl-N-[2-(naphthalen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(4-chlorophenyl)ethyl]-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
5-({8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)thiophene-3-carboxamide
N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
4-(2-{4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)morpholine
1-(3-fluorobenzoyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
methyl 1-[(3R,5S)-1-propyl-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-methanesulfonylpropan-1-one
3-cyclohexyl-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-pyrazole
1-[5-(2,6-difluoro-3-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-1-yl]butan-2-ol
2-({[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}(thiophen-3-ylmethyl)amino)butan-1-ol
3-benzyl-5-[(1R,2R)-2-phenylcyclopropyl]-1H-1,2,4-triazole
8-acetyl-2-[(4-fluoro-3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(5-methylfuran-2-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
2-butyl-8-[(6-chloropyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
6-[2-(5-fluoro-2-methoxyphenyl)-1H-imidazol-1-yl]-2-methylheptan-2-ol
1-[1'-(3-hydroxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-({3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-2-(propan-2-yl)-1H-imidazole
1-(naphthalen-2-yl)-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperazine
N-[2-(1-{3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanoyl}piperidin-2-yl)ethyl]acetamide
2-ethyl-4-phenyl-9-(1,3-thiazol-2-yl)-2,9-diazaspiro[5.5]undecane
3-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol
(2R,6R)-4-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(propane-1-sulfonyl)piperidine-3-carboxylate
N-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}methanesulfonamide
(4aR,7aS)-N,N-dimethyl-4-(2-methyl-1,3-thiazole-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-methoxy-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
2-cyclopropyl-8-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propyl}aniline
9-(2-methylbenzenesulfonyl)-3,9-diazaspiro[5.6]dodecane