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4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
({2-[(2-fluorophenyl)methoxy]-7-methoxyquinolin-3-yl}methyl)[2-(1H-imidazol-1-yl)ethyl]amine
3-(3-methoxyphenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-5-methyl-1H-pyrazole-3-carboxamide
methyl 4-{[3-(cyclopropylcarbamoyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}benzoate
1-(4-methyl-1,3-thiazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[2-(2-methoxy-5-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenoxy)ethyl]-2,1,3-benzothiadiazole-4-sulfonamide
N-[(2-chloropyridin-3-yl)methyl]-2-methoxy-N-methyl-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(1S,5R)-6-benzyl-3-{2-[4-(hydroxymethyl)phenyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
1'-[(3-fluoro-4-methoxyphenyl)methyl]-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]pyrimidin-2-amine
2-(4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}piperidin-1-yl)pyrimidine
1-butyl-5-(dimethyl-1,3-thiazol-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
N-[2-(3-chlorophenyl)ethyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(azocan-1-yl)-3-{5-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-2-methoxyphenoxy}propan-2-ol
1-(2-methylphenyl)-4-(1H-pyrazole-4-carbonyl)-1,4-diazepane
4-[4-(4-methoxyphenoxy)piperidin-1-yl]pyridine
6-amino-2-(2-{4-[2-(2-methylphenyl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)pyrimidin-4-ol
2-(1H-imidazol-2-yl)-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)benzamide
methyl(1,3-thiazol-2-ylmethyl)[(4-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
1-ethyl-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
2-(5-methyl-1,2-oxazole-3-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
N-[(1-benzylpyrrolidin-3-yl)methyl]-N-methyl-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
2-(5-methyl-1,2-oxazol-3-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidine
1-(6-methyl-2-phenylpyrimidin-4-yl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-(1-{7-[3-(1,3-benzothiazol-2-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
3-(2-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
2-[4-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)phenoxy]-1-(pyrrolidin-1-yl)ethan-1-one
6-chloro-4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}quinoline
1-{2-[(3S,4R)-3-cyclopropyl-4-{[6-(methoxymethyl)pyrimidin-4-yl]amino}pyrrolidin-1-yl]ethyl}pyrrolidin-2-one
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(1-methyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
4-(1H-pyrazol-1-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]piperidine-4-carboxylic acid
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-5-methyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-(4-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
8-benzyl-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-benzyl-5-[(furan-2-ylmethyl)(methyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-fluoro-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-(3-methylphenyl)pyrimidine
1-(3-methylfuran-2-carbonyl)-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
4-[(4-methyl-5-{[(2,2,3,3-tetrafluorocyclobutyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]piperidine
N,N-dimethyl-4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]piperazine-1-carboxamide
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
3-(4-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)-2,5-dimethylpyrazine