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1-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-N-(propan-2-yl)piperidine-4-carboxamide
6-methyl-1-[3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]-1,2-dihydropyridin-2-one
N-(2-methoxyethyl)-4-(piperidin-3-yl)-N-(pyridin-3-ylmethyl)benzamide
3-ethyl-5-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-1,2,4-oxadiazole
(3S,4R)-1-[2-(cyclopropylcarbamoyl)ethyl]-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-[5-(thiophen-2-yl)furan-2-yl]propan-1-one
2-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]aniline
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-N,N-dimethylazepan-4-amine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,4-diazepane
2-butyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-[2-(phenylsulfanyl)ethyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(furan-2-ylmethyl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(pyridin-2-ylmethyl)acetamide
(2,1,3-benzoxadiazol-4-ylmethyl)[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amine
({4-[(1-cyclohexanecarbonylpiperidin-3-yl)methoxy]phenyl}methyl)(methyl)(2-phenylethyl)amine
1-(cyclohexylmethyl)-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-6-oxopiperidine-3-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
2-{4-[(2,4-dimethoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
2-[4-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
4-({[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]amino}methyl)benzene-1-sulfonamide
1-(2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(4-acetyl-4-phenylpiperidin-1-yl)-3-(pyridin-2-yl)propan-1-one
2-methanesulfonyl-N-[(3-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)acetamide
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
2-(3,5-dichloropyridin-4-yl)-7-methyl-1H-1,3-benzodiazole
3-({[(1-ethylpyrrolidin-3-yl)methyl](methyl)amino}methyl)benzonitrile
N-(3-ethoxypropyl)-2-(N-phenylmethanesulfonamido)propanamide
N-(3-hydroxy-2,2-dimethylpropyl)-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-4-(piperidin-1-ylmethyl)benzamide
ethyl 2-{4-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]morpholin-3-yl}acetate
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-N-(pyridin-2-ylmethyl)pyridin-2-amine
2,3-dimethoxy-N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}benzamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(3-methylthiophene-2-carbonyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-3-phenyladamantane-1-carboxamide
1-{2-oxo-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}pyrrolidin-2-one
2-fluoro-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5-sulfamoylbenzamide
6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purine
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]pyridin-2-ol
1-tert-butyl-4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyrrolidin-2-one
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
2-[5-(5-amino-4-chloro-1H-pyrazol-3-yl)-1-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]acetamide
4-(1H-imidazol-1-ylmethyl)-1-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-ol
2-[4-(pyrimidin-2-yl)piperazin-1-yl]-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
3-(carbamoylmethoxy)-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
N-{1-[1-(1-carbamoylcyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
2-(4-ethylpiperazin-1-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
N-(3-{[(1-benzylpiperidin-4-yl)amino]methyl}-5-(pyrrolidine-1-carbonyl)phenyl)pyridine-2-carboxamide
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one