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1-(4-fluoro-2-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}phenyl)-3,5-dimethyl-1H-pyrazole
3-{[(3R)-piperidin-3-yl]sulfamoyl}-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
(5S,9aS,9bS)-5-(3-chloro-4-hydroxy-5-methoxyphenyl)-2-cyclopentyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-methoxy-N-[2-(1-methylpiperidin-3-yl)ethyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
2-(dimethylamino)-1-[4-(4-hydroxybutyl)piperazin-1-yl]-2-(4-methylphenyl)ethan-1-one
3-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,5-dimethoxyphenyl)methyl]piperidine
2-{4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
1-[4-(4-acetylphenyl)piperazin-1-yl]-3-[(3S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)piperidin-3-yl]propan-1-one
3-[(3R,4S)-1-(2,6-dimethoxypyridine-3-carbonyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
2-(5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl)acetamide
2-[5-(2-chlorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-ol
3-(1H-1,3-benzodiazol-2-yl)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}propanamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-3-methoxy-N-(oxolan-2-ylmethyl)benzamide
6-{[methyl(thian-4-yl)amino]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-hexanamidoacetic acid
3-(3-methylbutyl)-8-(quinoxaline-6-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-cyclohexyl-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]piperidine-4-carboxamide
2-(3-methyl-4-{[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
4-[4-(3-chloropyridin-2-yl)piperazine-1-carbonyl]-1-ethylpyrrolidin-2-one
3-(2-oxo-2-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}ethyl)-1,2,3-oxadiazol-3-ium-5-olate
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(phenylformamido)acetamide
1-(3-chloro-4-methylbenzoyl)-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-fluoro-5-sulfamoylbenzamide
1-[2-methoxy-5-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
(2S)-3-methyl-2-({1-[1-(3-phenylpropyl)piperidin-4-yl]piperidin-4-yl}formamido)butanamide
2-cyclobutyl-5-(2-methoxyacetamido)-1-methyl-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
3-[(1-ethylpiperidin-3-yl)methyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
1-(2-methanesulfonylethyl)-4-phenyl-5-(2-phenylethyl)-1H-imidazole
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(hydroxymethyl)piperidin-4-ol
(3aS,6aS)-2-cyclobutanecarbonyl-5-(2-phenoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1,6-dimethyl-3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
(2-methoxyethyl)[2-phenyl-1-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)ethyl](pyridin-3-ylmethyl)amine
1-(1-{[3-methoxy-4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
N-(3-cyclopentaneamido-4-methylphenyl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
propan-2-yl 2-chloro-5-{imidazo[1,2-a]pyridine-3-amido}benzoate
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidine-4-carbonitrile
N-[(3-chlorophenyl)methyl]-1-methyl-N-(2-methylpropyl)-1H-imidazole-2-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(propan-2-yl)amino]methyl}piperidin-2-one
3-{[cyclopropyl({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl})amino]methyl}phenol
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-acetyl-N,2,4-trimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrrole-3-carboxamide
1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-oxopyrrolidin-1-yl)propanamide