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3-{2-[2-(2-chloro-6-fluoro-3-methylphenyl)-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one
1-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
2-(butylsulfanyl)-N4-methyl-N4-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidine-4,6-diamine
4-methoxy-N-(2-methoxyethyl)-2-({1-[1-(5-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
1-benzyl-4-(6-methylpyridin-2-yl)-1,4-diazepan-6-ol
N-ethyl-5-[2-(3-methoxyphenyl)piperidine-1-carbonyl]pyrimidin-2-amine
3-phenyl-7-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]-1H-pyrazole-3-carboxylic acid
4-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydroisoquinolin-1-one
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
2-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-N-methyl-N-phenylacetamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
3-cyclopropyl-1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[(5-methylthiophen-2-yl)methyl]urea
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(2-methylphenyl)methyl]piperazin-2-one
(2S,4S)-4-{[(2,4-dimethoxyphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
4-(4-methylpyridin-3-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-methyl-7-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-oxo-1-{2-[(pyridin-3-yl)amino]ethyl}pyrrolidine-3-carboxylic acid
1-(2-chloro-6-methylbenzenesulfonyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
3-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)pyridin-2-amine
5-butyl-1'-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-[2-(1H-imidazol-1-yl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1-(2-methoxyethyl)-6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
N-[4-(pyridin-3-yloxy)phenyl]-2-(pyrrolidin-3-yl)benzamide
(3aR,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-N-cycloheptyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-5-methylpyrazine-2-carboxamide
N-[1-(3,5-difluorophenyl)cyclopropyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-hydroxy-N-[(3-hydroxypyrrolidin-3-yl)methyl]-3,5-bis(propan-2-yl)benzamide
(3S,4R)-3-ethyl-4-methyl-1-[3-(1H-1,2,4-triazol-1-yl)adamantane-1-carbonyl]piperidin-4-ol
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-8-fluoroquinoline-2-carboxamide
1,3-dimethyl 5-[4-(aminomethyl)phenyl]benzene-1,3-dicarboxylate
(3aR,6aR)-2-acetyl-N-[2-(2-fluorophenoxy)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(3aR,6aR)-2-[(5-propylfuran-2-yl)methyl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1,3,7-trimethyl-2-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1H-indole
1-[1'-(1-methyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-(1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazol-4-yl)phenol
1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
N-cyclopentyl-6-(5-methylpyridin-3-yl)pyridazin-3-amine
5-(methoxymethyl)-N-[(2-methoxyphenyl)methyl]-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N3-butyl-4-oxo-1-(propan-2-yl)-N5-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2,3,5-trimethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-methyl-6-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1,6-dihydropyridazine-3-carboxamide
N-{[4-(3-methoxyphenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclobutanecarboxamide
3-{5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}benzonitrile
5-[(2,3-dihydro-1H-inden-2-yl)amino]-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-hydroxyethyl)-N-methyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide