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3-(6-hydroxyhexyl)-N,N-dimethylbenzamide
1-[2-({6-[benzyl(methyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}amino)ethyl]piperidin-3-ol
(4aS,7aR)-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-6-{4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyrimidin-2-amine
4-{3-[2-(2-methoxyphenyl)-1H-imidazol-1-yl]propyl}-3,5-dimethyl-1H-pyrazole
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-methyl-1,4-diazepan-5-one
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2,6-dimethoxypyridine-3-carboxamide
3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole
3-[4-(9H-fluoren-2-yl)-1H-1,2,3-triazol-1-yl]propane-1,2-diol
N-ethyl-3-{[(4-methylphenyl)methyl]amino}-N-(pyridin-4-ylmethyl)benzamide
1-[3-(3-ethylphenoxy)azetidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]propan-1-one
(2S,4R)-4-[4-({[(3-chlorophenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-(2-cyclopropylpyrimidin-5-yl)-N,N,6-trimethylquinoline-4-carboxamide
2-oxo-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,2-dihydroquinoline-4-carboxamide
4-{1-[3-(dimethylamino)-1-phenylpropyl]-1H-imidazol-2-yl}benzoic acid
(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(1H-pyrrol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-({[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amino)-1-(2-phenylethyl)pyrrolidin-2-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-oxo-4H-chromene-2-carboxamide
1-(3-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
2-fluoro-4-(7-methyl-1H-indol-3-yl)phenol
(2S,4R)-1-(2-amino-6-methylpyrimidine-4-carbonyl)-N-ethyl-4-pentanamidopyrrolidine-2-carboxamide
(2S,4S)-N-ethyl-1-[2-(methylsulfanyl)acetyl]-4-[2-(pyridin-2-yl)acetamido]pyrrolidine-2-carboxamide
2-{[2-(oxan-3-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(3S,4S)-4-cyclopropyl-1-(4,5-dimethylthiophene-2-carbonyl)pyrrolidine-3-carboxylic acid
methyl (2S,4S,5R)-1,2-dimethyl-4-[methyl(pyridin-3-ylmethyl)carbamoyl]-5-phenylpyrrolidine-2-carboxylate
4-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-(2-phenylethyl)-5-(1-{6-[(propan-2-yl)amino]pyrimidin-4-yl}piperidin-4-yl)imidazolidine-2,4-dione
1-cyclopropyl-4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyrrolidin-2-one
4-benzyl-2-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
4-[4-(3,4-dimethoxyphenyl)-1H-imidazol-2-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
2-[(2-chlorophenyl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl[2-methyl-2-(morpholin-4-yl)propyl]{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-[(3R,4R)-3-[(4-ethylpiperazin-1-yl)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2,4-dimethylpyridine-3-carbonitrile
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}urea
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[3-(dimethylamino)propyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
2-(dimethylamino)-N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-(3-methylphenyl)acetamide
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-[(5-ethylpyridin-2-yl)methyl]urea
{2-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-1-(furan-2-yl)ethyl}diethylamine
{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidin-4-yl}methanol
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-amine
1,3-dimethyl-N-[2-(morpholin-4-yl)butyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
(3ar,6ar)-N-{[1-(methoxymethyl)cyclopentyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2,4-dimethoxy-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
(3R,4R)-4-amino-1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-3-ol
1-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
5-fluoro-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1H-indole