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2-methyl-7-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-methyl-4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-2-one
2-hydroxy-3-(2-methylphenoxy)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]propanamide
3-benzyl-1-methyl-8-[3-(5-methylfuran-2-yl)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
methyl(1,2-oxazol-5-ylmethyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
(2S,4S)-4-amino-1-[3-(3-methoxyquinoxalin-2-yl)propanoyl]-N-methylpyrrolidine-2-carboxamide
3-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-N-methylpyridin-2-amine
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
3-cyclopropyl-1-[4-(furan-2-ylmethoxy)phenyl]-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
N3-(adamantan-1-ylmethyl)-1-cyclopentyl-N5,N5-diethyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-2-yl)pyridine
2-[2,6-dimethyl-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-methoxypyrazine
(1R,3S)-3-(2-aminoethoxy)-7-(2,3-dihydro-1H-indene-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
4-{3-[(3S)-3-ethylmorpholine-4-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
N-[2-(4-methoxyphenyl)ethyl]-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-cyclohexyl-4-{thieno[2,3-d]pyrimidin-4-yl}piperazin-2-one
5-chloro-N-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
3-(2,4-dimethoxybenzoyl)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidine
5-ethyl-N4-methyl-N4-[2-(oxan-2-yl)ethyl]pyrimidine-2,4-diamine
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-[(2-chlorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
3-(1-{2-[(4-methylphenyl)sulfanyl]ethyl}-1H-1,2,3-triazol-4-yl)phenol
2-chloro-4-({cyclopropyl[(2-ethoxyphenyl)methyl]amino}methyl)-6-methoxyphenol
4-(3-benzyl-1H-pyrazol-5-yl)-1-(1H-imidazol-4-ylmethyl)piperidine
2-(2,2-dimethylpropanamido)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-methylthiophene-3-carboxamide
1-{2-[1-(1-methylpiperidin-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
(4aS,7aR)-1-(2-fluorobenzenesulfonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-2-yl}-1,3-benzothiazole
(2S,4S)-4-amino-N,N-diethyl-1-[2-(4-fluoro-3-methylphenyl)acetyl]pyrrolidine-2-carboxamide
1-{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-4-yl}-3-phenylpropan-1-ol
(2S,4S)-4-amino-N,N-diethyl-1-[3-(4-fluorophenyl)propanoyl]pyrrolidine-2-carboxamide
N-(2,4-dimethoxyphenyl)-3-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]propanamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-1-(2-methoxyethyl)pyrrolidin-2-one
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-(1H-imidazol-1-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
2-{4-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]phenyl}ethan-1-amine
2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]ethan-1-one
4-(1H-imidazol-1-yl)-1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
2-(2-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
2-fluoro-5-sulfamoyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]benzamide
5-(3-{6-azabicyclo[3.2.1]octan-6-yl}-3-oxopropyl)-5-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-1,4-dimethylpiperidine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-1,2,3-thiadiazole-5-carboxamide
4-(2-aminoacetyl)-5-butyl-1-(3-phenylphenyl)piperazin-2-one
(3S,7S)-5-(oxane-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
1-[benzyl(methyl)amino]-3-{2-methoxy-5-[(4-propylpiperazin-1-yl)methyl]phenoxy}propan-2-ol