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N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-amine
2-methoxy-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
1-[2-(dimethylamino)ethyl]-5-(2-hydroxy-4-methylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3S)-3-({[3-chloro-5-ethoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)azepan-2-one
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)morpholine-4-sulfonamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
(3R,4R)-3,4-dimethyl-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-ol
2-(2,3-difluorophenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,3-oxazole-4-carboxamide
5-[1-(3-methylfuran-2-carbonyl)pyrrolidin-2-yl]-N-(1,3-thiazol-2-yl)thiophene-2-carboxamide
N-cyclopropyl-1-(1-methylpiperidin-4-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxamide
2-(1-cyclopentyl-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl)ethan-1-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
(1-{[(5,6-dimethylpyrimidin-4-yl)(methyl)amino]methyl}cyclopentyl)methanol
(2S,4S)-4-amino-1-(2,6-dimethoxypyridine-3-carbonyl)-N-ethylpyrrolidine-2-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
4-{4-[2-(methylsulfanyl)benzoyl]piperazin-1-yl}quinazoline
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]quinoline
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[4-(diethylsulfamoyl)phenyl]-N-ethylbenzamide
N,1,6-trimethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{[2-(diethylamino)ethyl]amino}-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
2-(1H-imidazol-1-yl)-N-{[3-methyl-7-(5-phenoxyfuran-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}acetamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(3S)-N,N-dimethyl-1-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}azepan-3-amine
3-[4-(pyridin-4-yl)piperazine-1-carbonyl]-5,6,7,8-tetrahydroquinoline
N-methyl-N-(1,2-oxazol-5-ylmethyl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-chloro-5-({3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
N,N-dimethyl-5-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
methyl[(2-phenyl-1,3-thiazol-4-yl)methyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-ol
4-ethyl-5-methyl-6-{3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}pyrimidin-2-amine
N-({1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]pyrrolidin-3-yl}methyl)methanesulfonamide
1-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-5-phenylpentan-1-one
2-(2,3-dimethylphenyl)-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}acetic acid
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyridine
2-(3,4-dichlorophenyl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
(1S)-1-[3-(cyclopropylmethyl)-1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethan-1-amine
3-chloro-5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-(2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-fluoro-5-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]benzonitrile
4-methyl-5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyrimidine
1-(2,5-dimethylfuran-3-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
ethyl 4-(oxan-2-ylmethyl)-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine-4-carboxylate
N-cyclohexyl-1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
2-(pyridin-2-yl)-5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]pyrimidin-4-ol
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-ol
1-[1-(5-acetylpyridin-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
2-chloro-4-({[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)phenol