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(4S)-N-(cyclohexylmethyl)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carboxamide
(2R)-2-amino-N-[(5-ethylpyridin-2-yl)methyl]-N,4-dimethylpentanamide
N-[(3S,4R)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
1-[2-methoxy-4-({[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-(2,3-dihydro-1H-inden-2-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[(3R,4R)-3-hydroxy-1-(3-hydroxypyridine-2-carbonyl)piperidin-4-yl]pyridine-3-carboxamide
3-(oxolan-3-yl)-5-[(4,6,7-trimethyl-1-benzofuran-3-yl)methyl]-1,2,4-oxadiazole
1-cyclopentanecarbonyl-3-(2-methoxyphenoxy)azetidine
2-methyl-8-(piperidine-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-methyl-3-[N-methyl-1-(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]butanamide
(3R,4S)-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3,4-dimethylpiperidin-4-ol
1-(hexan-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{1-[1-(2-methoxy-2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(2R,6R)-11-methoxy-4-(pyridin-2-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{2-methyl-4-[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
[1-(2-fluorophenyl)propan-2-yl][3-(4-methyl-1H-pyrazol-1-yl)propyl]amine
1-{1'-[(4-chloro-3-fluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2,2-dimethyl-N-{1-[1-(1-propylpiperidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
3-(2-methoxyethyl)-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,2,4-oxadiazole
5-{[benzyl(methyl)amino]methyl}-N-[(2,5-dimethylphenyl)methyl]-1,2-oxazole-3-carboxamide
2-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-({1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
4-(4-methoxy-2-methylphenyl)-3-(2-methyl-1,3-oxazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-2-(4-methyl-1H-pyrazol-1-yl)acetamide
8-cyclopropanecarbonyl-2-(2,5-dimethylfuran-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-hydroxy-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-(3-chloro-4-fluorophenyl)-3-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}propanamide
1-{2-[(3R,4S)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]ethyl}pyrrolidin-2-one
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(methoxymethyl)piperidine
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-ethoxyphenoxy)ethyl]methylamine
N,2-dimethyl-N-[3-(oxolan-2-yl)propyl]thieno[3,2-d]pyrimidin-4-amine
2-(4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}morpholin-3-yl)acetic acid
2-methoxy-1-{4-[(2-phenylphenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
N-methyl-2-(3-{3-[6-(piperidin-1-yl)pyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)acetamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]benzamide
3-(4-fluorophenyl)-5-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-{1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
(4aS,8aR)-1-(3-hydroxypropyl)-6-(1-phenylcyclopropanecarbonyl)-decahydro-1,6-naphthyridin-2-one
1-[(1S,5R)-6-(5-chloro-3-methyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
6-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(3,4-dimethoxyphenyl)propan-1-one
2,3,6-trifluoro-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
5-(azepane-1-carbonyl)-N-[furan-2-yl(phenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N,N-dimethyl-5-[3-(1-methylpiperidin-3-yl)propanoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-pyrazole-4-carboxamide
N-[4-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-oxobutyl]acetamide
6-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
N-[(3R,4R)-1-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
4-(2,5-dimethoxybenzoyl)-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide