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{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1,3-thiazol-4-yl)ethyl]amine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
1-benzyl-5-{[(2,3-difluorophenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2-hydroxyethyl)-8-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}pyridine-3-carboxylic acid
2-{4-[(6-ethylpyrimidin-4-yl)amino]piperidin-1-yl}ethan-1-ol
4-{[4-(furan-2-yl)phenyl]methyl}-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1s,4s)-4-[3-(2-hydroxyphenyl)-1H-pyrazole-5-amido]cyclohexane-1-carboxylic acid
(2S,4S,5R)-5-(2-fluorophenyl)-4-[(1H-imidazol-2-ylmethyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
1-methyl-4-({4-methyl-5-[1-(propan-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
3-(3,4-dimethylphenyl)-N-methyl-N-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
4,5-dimethyl-6-[4-(oxolan-3-ylmethyl)piperazin-1-yl]pyrimidine
1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}azetidin-3-ol
N-[2-(1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)ethyl]acetamide
(2S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-methyl-2-phenylpiperazine
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(pyrrolidin-3-yl)acetamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-(3-{[3-(3-methylphenyl)phenyl]carbamoyl}piperidine-1-carbonyl)pyridin-1-ium-1-olate
1-[(2-aminopyridin-3-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
6-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-(5-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
2-(4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)pyridine-3-carbonitrile
N-(furan-2-ylmethyl)-4-(4-methylpiperazin-1-yl)-N-(prop-2-yn-1-yl)benzamide
1-[(4-fluorophenyl)methyl]-N-[2-(pyrazin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-{4-[5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl]piperazin-1-yl}phenol
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
9-[3-(methylsulfanyl)propyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2,2-dimethyl-5-[4-(2-phenylethyl)piperidine-1-carbonyl]thiomorpholin-3-one
7-fluoro-N-(5-methanesulfonyl-2-methylphenyl)-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-(propan-2-yl)piperazine
2-(dimethylamino)-2-(4-methylphenyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(dimethylamino)acetamide
2-(6-aminopyridin-3-yl)-2-{methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amino}acetic acid
4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-(2-phenylethyl)piperazin-2-one
2-(morpholin-2-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)acetamide
2-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-1,3-thiazole-4-carboxamide
1-[(4-methanesulfonylphenyl)methyl]-2-(2-methoxyphenyl)pyrrolidine
N-(1H-imidazol-2-ylmethyl)-N,5,6-trimethylthieno[2,3-d]pyrimidin-4-amine
N-methyl-N-(pyridin-2-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
9-[(2E)-3-phenylprop-2-en-1-yl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-(2-aminoethyl)-6-{pyrazolo[1,5-a]pyridine-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
2-(adamantan-1-yl)-N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)acetamide
N-cyclopentyl-4-(9H-fluoren-2-ylmethyl)morpholine-2-carboxamide
(2S,4S)-4-amino-1-{2-[(3-methoxyphenyl)sulfanyl]acetyl}pyrrolidine-2-carboxylic acid
ethyl 5-{methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylate
1-[(3-chloro-4-propoxyphenyl)methyl]-3-[(dimethylamino)methyl]piperidin-3-ol
(2S,4R)-4-amino-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylpyrrolidine-2-carboxamide
N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
6-[(3-fluorophenyl)methoxy]-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one