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2-[2-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)-4-(pyrimidin-2-yl)phenoxy]acetic acid
2-amino-4-(3-ethoxy-4-hydroxyphenyl)-6-hydroxy-5H-indeno[1,2-b]pyridine-3-carbonitrile
(1S,5R)-3-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-phenyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,2-oxazole-3-carboxamide
2-(pyridin-2-yl)-6-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
N-(1-{1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
5-{[4-(1H-imidazol-2-yl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
diethyl({[3-(morpholine-4-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
3-[2-(2,6-difluorophenyl)ethyl]-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine
7-chloro-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
(3R,5S)-N3-(4-fluorophenyl)-N5-(3-methoxypropyl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
2-({3-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})carbamoyl]phenyl}amino)acetic acid
6-(dimethylamino)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-methoxy-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydropyridin-2-one
N-(2-hydroxyethyl)-1-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-(cyclohexylmethyl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}piperidin-2-one
2-acetyl-8-(oxan-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(2-{methyl[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)piperidin-2-one
5-chloro-3-methyl-2-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1H-indole
1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
(4aS,8aS)-2-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
4-(3-hydroxy-3-methylbutyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)benzamide
7-(2-methylphenyl)-4-(pyridazine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{[2-hydroxy-3-(3-methoxyphenoxy)propyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[1-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(morpholin-4-yl)ethyl]-3-(piperidin-4-ylmethyl)benzamide
(2R,3R,6R)-3-phenyl-5-[3-(1H-pyrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-({[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
(2S,4S,5R)-5-(2-chlorophenyl)-4-[(2-hydroxyethyl)(methyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylic acid
3-(2-chlorophenyl)-1-methyl-6-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(2-methyl-1-benzofuran-7-yl)-4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-carboxamide
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-pyrazol-3-yl)benzamide
(3S,4S)-1-(2-{[(4-chlorophenyl)methyl]carbamoyl}ethyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
(3R,5R)-5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]pyrrolidin-3-ol
4-(4-acetyl-4-phenylpiperidin-1-yl)-4-oxobutane-1-sulfonamide
2-(4-fluorophenyl)-2-(piperidin-1-yl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one
2-{2-[(E)-2-phenylethenyl]phenyl}ethan-1-amine
6-[4-(piperidine-1-carbonyl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
11-{[(2-chlorophenyl)methyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(dimethylamino)-N-(1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-phenylethyl)-N-methylacetamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-(3,4-dimethoxyphenyl)ethyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
8-(1H-indol-2-ylmethyl)-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(2-fluorophenoxymethyl)piperidine
2-amino-4-(3-chloro-5-fluoro-4-methoxyphenyl)-6-(pyridin-2-yl)pyridine-3-carbonitrile
2-[4-(hydroxymethyl)phenyl]-2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]acetic acid