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2-[3-(dimethylamino)propyl]-9-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
(3aS,6aR)-N-butyl-3-[(3,4-dimethoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
1'-[1-(propan-2-yl)-1H-pyrazole-5-carbonyl]spiro[indene-1,4'-piperidine]
(3S,4S)-4-propyl-1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidine-3-carboxylic acid
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-fluorobenzamide
N-methyl-N-(2-methylprop-2-en-1-yl)-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
1-{[(2S,4S)-1-[3-(2,3-dihydro-1H-indol-1-yl)propanoyl]-4-fluoropyrrolidin-2-yl]methyl}-3,3-dimethylurea
N-{[1-(2,3-dihydro-1H-inden-5-yl)-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl]methyl}acetamide
1-cyclopropyl-4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-2-one
7,7-dimethyl-2-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(1-cyanocyclopropanecarbonyl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
(3R,4R)-1-{[2-(cyclopentyloxy)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
1-[cyclohexyl(methyl)amino]-3-[2-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-methyl-1H-indole
4-(cyclopropylmethyl)-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
[(4-methoxyphenyl)methyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})(pyridin-4-ylmethyl)amine
{1-[(1-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
3-{[(furan-2-ylmethyl)(1-hydroxybutan-2-yl)carbamoyl]amino}-N,2-dimethylbenzamide
N,2-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-3-(1H-pyrazol-1-yl)propanamide
2,4-dichloro-6-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}phenol
N,N-dimethyl-3-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazin-2-amine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
2-methoxy-4-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
4-(3,4-difluorobenzoyl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperidine
1-cyclohexanecarbonyl-N-[2-(piperidin-1-yl)ethyl]pyrrolidine-2-carboxamide
4-methyl-2-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
2-(2,4-difluorophenoxy)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]acetamide
1-(furan-2-ylmethyl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]piperidine-4-carboxamide
1-(2-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}pyrimidin-4-yl)piperidin-3-ol
1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(2-methoxyphenyl)-2-methyl-1-(6-methylpyridine-2-carbonyl)piperazine
1-(2-cyclohexylethyl)-3-hydroxy-3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)piperidin-2-one
N-[(3R,4S)-1-(2-ethoxyethyl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
4-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
4-hydroxy-N-methyl-N-[2-(phenylsulfanyl)ethyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
[(5-chlorofuran-2-yl)methyl][(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}-2,6-dimethylphenol
2-(1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
4-[4-(4-methylphenoxy)piperidine-4-carbonyl]morpholine
N-(4-butylphenyl)-4-(morpholin-4-yl)piperidine-1-carboxamide
{1-[1-(2-ethoxypyridine-3-carbonyl)piperidin-3-yl]piperidin-4-yl}methanol
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-N-methylpyridin-2-amine
4-[2-(piperidine-1-carbonyl)phenoxy]-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
5-(4-methyl-3-phenylpiperazine-1-carbonyl)-1H-indole
2-[3-(2-methoxyethyl)-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
N3-[1-(2-chlorophenyl)ethyl]-N5-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide