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3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-({4-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-3-methoxyphenyl}methyl)piperazine-1-carboxamide
N-[1-(pyrazin-2-yl)propan-2-yl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
4-{3H-imidazo[4,5-b]pyridin-5-yl}-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-4-ylmethyl)amino]ethyl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
4-(2-phenylethyl)-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-amino-2-methyl-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
2-[2-(1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
N-(butan-2-yl)-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(pyridin-4-ylmethyl)benzamide
1-methyl-3-(2-{[(4-methylphenyl)methyl]sulfanyl}phenyl)-1-(oxan-4-yl)urea
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(1-butyl-4-methyl-1H-pyrazol-5-yl)butanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
8-methoxy-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)propanamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(1-benzyl-3-oxopiperazin-2-yl)acetamide
2,3-dimethyl-7-(pyridine-3-sulfonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-7-methyl-1-benzofuran-2-carboxamide
6-[(3R,4S)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-4-(1H-1,2,4-triazol-1-yl)butanamide
N-(4-methoxy-2-methylphenyl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-2-yl)piperazine
N3-benzyl-N5-[(4-methoxyphenyl)methyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-[(4-methylphenyl)methyl]-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
2,2-difluoro-N-[2-(4-phenylpyrimidin-2-yl)ethyl]propanamide
propyl 4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
4-[5-(methoxymethyl)furan-2-carbonyl]-1-(4-methylphenyl)piperazin-2-one
8-{[2,5-dimethyl-1-(pyridin-3-ylmethyl)-1H-pyrrol-3-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-imidazol-2-yl}pyridine
2-methyl-6-[2-(oxane-4-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
3-{[(2-carbamoylethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(2S)-2-acetamido-N-ethyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}propanamide
(benzylsulfamoyl)[4-(pyridin-2-yl)butyl]amine
2-(3-methoxypropyl)-8-(7-methyl-1-benzofuran-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(2E)-1-{3-[5-(2-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl}-3-(3,4-difluorophenyl)prop-2-en-1-one
methyl 1-cyclohexyl-2-oxo-3-(pyrimidin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]butan-1-one
ethyl 1-(2,5-dimethoxybenzoyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
N,N-dimethyl-4-[4-(2-methylphenyl)piperazin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]benzamide
7-cyclopropanecarbonyl-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(adamantan-1-yl)-5-(2-butylpyrrolidine-1-carbonyl)pyrimidin-4-ol
4-{4-[(dimethylamino)methyl]thiophen-2-yl}-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-methyl-6-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
(1S,5R)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[1-(2-acetamidoacetyl)piperidin-3-yl]benzoic acid