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2-(3-methyl-1H-pyrazol-1-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)acetamide
4-(1H-imidazol-1-ylmethyl)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
methyl (2S,4R)-4-acetamido-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
(3aR,6aR)-2-[(4-methyl-1H-imidazol-2-yl)methyl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-1-(2,3-dihydro-1-benzofuran-7-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-cycloheptyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
6-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridin-3-ol
2-(2,5-dioxoimidazolidin-4-yl)-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)acetamide
6-{[(7-chloro-4-methylquinolin-2-yl)amino]methyl}-2-methylpyrimidin-4-ol
3-{[6-oxo-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-{[(cyclohexylmethyl)amino]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-amino-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methylpropanamide
N-[3-(methylsulfanyl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
(2S)-1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-methyl-2-phenylpiperazine
1-[2-(4-fluorophenoxy)phenyl]-3-(3-hydroxy-2,2-dimethylpropyl)-3-methylurea
3-(4-hydroxyphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]propan-1-one
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]cyclohex-1-ene-1-carboxamide
(3R,9aR)-3-benzyl-8-(3,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2S)-1-[6-(benzyloxy)-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl]-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
N-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-1-(morpholine-4-carbonyl)piperidin-4-amine
N-[3-(benzyloxy)-2-hydroxypropyl]-5-phenyl-1,2-oxazole-3-carboxamide
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[(1-ethylpyrrolidin-2-yl)methyl]-2-oxo-3-(1,3-thiazol-4-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
7-[(2,3-dimethoxyphenyl)methyl]-2-(3-methoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-1,3-thiazole-4-carboxamide
2-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-{[1-(2-methylpropyl)piperidin-4-yl]amino}-N-(propan-2-yl)acetamide
5-acetyl-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-2,4-dimethyl-1H-pyrrole-3-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-4-[(4-methylpyrimidin-2-yl)amino]pyrrolidin-2-one
N,N-dimethyl-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]azepan-4-amine
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[3-(azepan-1-yl)-2-hydroxypropyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
3-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(quinoxaline-6-carbonyl)pyrrolidin-3-yl]urea
2-{[4-(pyrrolidine-1-sulfonyl)-1,4-diazepan-1-yl]methyl}-1H-1,3-benzodiazole
methyl (2S,4R)-4-hydroxy-1-({3-[(3-methylpyridin-2-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxylate
3-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}furan-2-carboxamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
(3E)-5,5-dimethyl-2-[4-(pyridin-4-yl)piperazin-1-yl]hex-3-enoic acid
1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-({3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}methyl)-6-ethoxyphenol
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
1-butyl-4-[(5-ethylfuran-2-yl)methyl]piperazin-2-one
N-[(6-chloropyridin-3-yl)methyl]-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(1R,7S)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide