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(2S,4S)-N-ethyl-4-[(naphthalen-1-ylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-[4-(benzylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(methylsulfanyl)ethan-1-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-{1-[3-(cyclohexyloxy)-2-hydroxypropyl]-1H-1,2,3-triazol-4-yl}phenol
N-cyclopentyl-3-{[(1-ethyl-1H-imidazol-5-yl)methyl]sulfamoyl}benzamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(3,5-dichlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(furan-2-yl)propyl]-3-azaspiro[5.5]undecan-9-amine
2-(3-{[2-(4-fluorophenyl)morpholin-4-yl]methyl}phenoxy)acetic acid
2-[4-(cyclopropylmethyl)piperazin-1-yl]-2-[4-(hydroxymethyl)phenyl]acetic acid
2-(3-methoxyphenyl)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
4-methoxy-1-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(prop-2-en-1-yl)piperidine
ethyl 4-(2-methoxyethyl)-1-[3-(5-methylfuran-2-yl)butyl]piperidine-4-carboxylate
N-[3-(methylsulfanyl)propyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
8-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
5-{2-[3-cyclopropyl-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}-1H-1,2,3,4-tetrazole
3-(2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-1-propyl-1H-pyrazole-5-carboxamide
1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-(3-methylthiophen-2-yl)-1-[(3,4,5-trimethoxyphenyl)methyl]-1H-imidazole
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[(6-methylpyridin-2-yl)methyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(2-acetylbenzoyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{1-benzyl-2-methyl-7-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methylpropanamide
4-fluoro-3-methoxy-N-methyl-N-[2-(pyridin-4-yl)ethyl]benzamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
N-(2-hydroxyethyl)-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
4-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]benzonitrile
1-(diethylamino)-3-[2-methoxy-4-({[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
(4aR,7aS)-1-benzyl-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-N-(pyridin-2-ylmethyl)acetamide
1-methyl-4-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]piperazin-2-one
2,3-dimethyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)quinoxaline-6-carboxamide
(2S,4S)-4-amino-1-(3-ethoxypropanoyl)-N,N-diethylpyrrolidine-2-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
(4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-2-yl)methanamine
N-[(3R,4S)-1-[(4-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxy-2-methylpropanamide
N5-tert-butyl-1-cyclohexyl-N3-methyl-N3-[(1-methylpiperidin-3-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl (2S,4S)-4-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-amido]-1-methylpyrrolidine-2-carboxylate
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
4-[2-(4-chlorophenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(2-hydroxy-2-phenylethyl)acetamide
1-({1-[1-(propane-2-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)azepane
4-(cyclopropylmethyl)-1-[2-(3-hydroxyphenyl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
methyl 3-[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)carbamoyl]propanoate
1-[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
5-[2-(pyridin-3-yl)-1H-imidazol-1-yl]-2,3-dihydro-1H-inden-1-one
1-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]-4-ethyl-1,4-diazepan-5-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide