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6-[(diethylamino)methyl]-N-(3-fluoro-4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one
3-(2,1-benzoxazol-3-ylformamido)-N-(2-fluoro-4-methylphenyl)propanamide
N-[(3S,4R)-1-(2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
N-[4-(4-{[1-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
2-amino-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-methylpropan-1-one
1-[3-({[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-(benzenesulfonyl)-4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
(3S,4S)-1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
2,2-dimethyl-N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]oxane-4-carboxamide
3-({methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
6-[(2-hydroxyethyl)(methyl)amino]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
(3R,4R)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-cyclobutyl-3-methylpiperidin-4-ol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-N-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
methyl 2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-1,3-benzodiazole-6-carboxylate
1-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-(5-chloro-2-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-{5-[2-(2-methoxyphenyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-[1-(adamantane-1-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-{3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]phenyl}imidazolidin-2-one
N-[(2,4-dimethoxyphenyl)methyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1R,5R)-6-(2-methoxyethyl)-3-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
6-(2H-1,3-benzodioxol-5-ylmethyl)-3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
4-{[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]formamido}-N,N-dimethylbutanamide
[(3R,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[2-(3-hydroxypiperidin-1-yl)ethyl]propanamide
4-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]morpholine
N-({1-[3-(2-acetamidopropyl)-1H-indole-2-carbonyl]piperidin-4-yl}methyl)acetamide
3-{[4-(2-amino-5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}phenol
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-N-[(2S)-2-hydroxypropyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2S)-3-methyl-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)butanamide
1-phenyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
2-[4-(2-fluorophenyl)piperazin-1-yl]-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
1-tert-butyl-N,N-bis(1,3-oxazol-4-ylmethyl)-5-oxopyrrolidine-3-carboxamide
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-2-propyl-2,5-dihydro-1H-pyrrole
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydroisoquinolin-1-one
N-(1-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1,4-diazepane
3-({[2-(2-methoxyethoxy)phenyl]carbamoyl}amino)-N,N-dimethylpropanamide
4-[4-(4,4-difluoropiperidin-1-yl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl]pyridine
1-[(4-fluorophenyl)methyl]-4-(5-methyl-1,2-oxazole-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
1-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
5-{1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-2-yl}-3-phenyl-1,2,4-oxadiazole
4-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-5-(propan-2-yl)pyrimidine
ethyl 1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate