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3-(propoxymethyl)-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrrolidine
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
1-(2,3-dihydro-1-benzofuran-2-ylmethyl)-3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methylurea
7-chloro-1-(3-hydroxypyrrolidine-1-carbonyl)-9H-fluoren-9-one
2-(3-fluoro-4-hydroxyphenyl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]ethan-1-one
methyl 3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)benzoate
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(1-benzyl-1H-pyrazole-4-carbonyl)-N-(4-methoxyphenyl)piperidin-3-amine
3-(2-methoxybenzoyl)-1-(4-methylbenzenesulfonyl)piperidine
4-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
4-(2-amino-6-hydroxypyrimidin-4-yl)-7-(3,6-dimethylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(pyridin-4-yl)ethan-1-ol
7-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}phenyl)benzenesulfonamide
N-ethyl-3-{[(2-methoxyethyl)(1-methylpiperidin-4-yl)carbamoyl]amino}-2-methylbenzamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(1H-imidazol-2-ylmethyl)acetamide
2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinolin-5-ylmethyl)acetamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
(3S,4S)-4-methyl-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidine-3,4-diol
(5-{1-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-imidazol-2-yl}furan-2-yl)methanol
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-[(2S)-4-methyl-1-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-1-oxopentan-2-yl]acetamide
[(8-chloroquinolin-2-yl)methyl](1,4-dioxan-2-ylmethyl)methylamine
1-[(1R,5R)-6-{[4-(2-hydroxyethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
7-[(4-fluorophenyl)methyl]-2-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
N-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}-4-(1H-pyrazol-3-yl)piperidine-1-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-7-fluoro-N,2-dimethylquinoline-4-carboxamide
3-[(3R,4S)-1-[(2-ethylphenyl)carbamoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
methyl 2-{[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazol-4-yl]formamido}acetate
2-(4-fluorophenyl)-1-(3-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxymethyl}piperidin-1-yl)ethan-1-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
[(2-ethylpyrimidin-4-yl)methyl](methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyridine-4-carboxamide
4-{5-[(3-methyl-3-phenylpiperidin-1-yl)methyl]pyrimidin-2-yl}morpholine
1-(6-cyclopropylpyrimidin-4-yl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
[(2S,6S)-4-[(2,4-dichlorophenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(3-methoxyphenoxymethyl)piperidine
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(2-chlorophenyl)-2-hydroxyethan-1-one
4-(4-acetyl-4-phenylpiperidin-1-yl)-1-phenylbutan-1-one
(1S,5R)-3-[(4-chlorophenyl)methyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-ethyl-5-({[3-(methylcarbamoyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-acetyl-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
(2S,4S)-4-{[(3,4-dimethoxyphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
N-cyclobutyl-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
8-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)pent-4-en-1-one
N,N-dimethyl-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonamide
[(3S,5R)-1-(furan-2-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)propanamide