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1-(5-propylthiophene-3-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
{5-[(2E)-3-phenylprop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-(2-methoxyethyl)-1,1-dioxo-N-(pyridin-4-ylmethyl)-1λ6-thiolane-3-carboxamide
N-propyl-2-[3-(1H-pyrazol-3-yl)phenyl]pyridine-3-carboxamide
4-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methoxypyrimidine
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-methoxyphenol
1-(2,3-dihydro-1H-inden-2-yl)-4-[(2,2-dimethyloxan-4-yl)methyl]piperazine
3-[(1-methyl-1H-imidazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
N-[1-(1-{3-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-methyl-N-(2-phenylethyl)piperidin-3-amine
7-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
2-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1-(3-methoxypropyl)-1H-imidazole
1'-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(3-chloro-1,2-oxazol-5-yl)-1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]propan-1-one
methyl 3-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-5-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)benzoate
1-({5-[1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-2,4-dimethylphenyl}methyl)-1H-1,2,4-triazole
2-ethyl-9-(1H-imidazol-2-ylmethyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(3R,5S)-5-(3-fluorophenoxymethyl)-N-(3-methoxypropyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
1-methyl-4-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-6-propyl-1H-pyrazolo[3,4-d]pyrimidine
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
(2S)-2-[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]pyrrolidine-1-carboxamide
2-[(3-methoxyphenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]morpholine
2-methoxy-3-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrazine
4-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-1-(cyclopropylmethyl)-2-(propan-2-yl)-1,4-diazepane
2-{4-cyclohexyl-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(4-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenoxy)pyrimidine
2-(dimethylamino)-2-(2-methylphenyl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
1-(2-fluorophenyl)-5-[(oxolan-2-ylmethoxy)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
5-cyclobutyl-N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-1,3,4-oxadiazol-2-amine
1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-[(3,4,5-trimethoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-{1-[3-(2-methylphenoxy)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-hydroxy-2-methyl-N-{3-[methyl(phenyl)amino]propyl}pyrimidine-5-carboxamide
2-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}benzonitrile
3-({[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-N'-phenylethanediamide
2-(2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-2-yl}ethyl)pyridine
N-(3-chloro-4-propanamidophenyl)-2-[(propan-2-yl)amino]benzamide
N-[(3R,4S)-1-acetyl-4-phenylpyrrolidin-3-yl]piperidine-1-sulfonamide
4-{2-oxo-2-[3-(propoxymethyl)pyrrolidin-1-yl]ethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-[(2-methyl-1H-imidazol-4-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
ethyl 2-[4-({[1-(pyridin-3-yl)propan-2-yl]carbamoyl}amino)phenyl]acetate
N-(butan-2-yl)-6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
[1-(1-benzylpyrrolidin-3-yl)-4-[(3-methoxyphenyl)methyl]piperidin-4-yl]methanol
N-ethyl-N-methyl-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-amine
4-(3,4-diethoxyphenyl)-2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazole
3-(2-phenylethyl)-7-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
8-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one