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2-{1-benzyl-4-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetic acid
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
4-[1-(3,4-difluorophenyl)piperidin-4-yl]-2-(trifluoromethyl)morpholine
(1H-imidazol-4-ylmethyl)(methyl){[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
5-fluoro-N-(2-methoxyethyl)-1-methyl-N-(thiophen-3-ylmethyl)-1H-indole-2-carboxamide
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)-4-(trifluoromethyl)benzamide
8-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)-N-methylpropanamide
4-[2-(2-aminoethyl)phenyl]-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-amino-4-[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
ethyl 1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
5-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
3-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
1-(cyclohexylmethyl)-N-(1H-indol-2-ylmethyl)-6-oxopiperidine-3-carboxamide
3-{2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-fluorophenoxymethyl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
1-ethyl-3-(morpholine-4-carbonyl)-5-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
(1S,5R)-3-(2-methyl-1,3-benzoxazole-6-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{[(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)amino]methyl}pyrrolidin-3-ol
5-propyl-1'-(2-propyl-1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-N-(quinolin-5-ylmethyl)-2,3-dihydro-1-benzothiophene-2-carboxamide
1-methyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclopropanecarboxamide
3-methyl-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)but-2-enamide
2-(2H-1,3-benzodioxol-5-yl)-1-(4-phenyl-1,4-diazepan-1-yl)ethan-1-one
3-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
2-amino-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)pyridine-4-carboxamide
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]acetamide
(4aS,7aR)-1-(furan-2-carbonyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-phenyl-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1,2,3,6-tetrahydropyridine
4-({[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]amino}methyl)hepta-1,6-dien-4-ol
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(thiophen-2-ylmethyl)propanamide
4-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]-1,3-dimethylpiperazin-2-one
2-ethyl-4-phenyl-9-(1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecane
4-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}morpholine
(3S,4R)-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
5-butyl-1'-(1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(propan-2-yl)acetamide
8-fluoro-2-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)quinolin-4-ol
(2S,4R)-1-[(2,5-dimethoxyphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-cyclopropyl-6,6-dimethyl-5-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]thiomorpholine-3-carboxamide
(2S)-2-{[4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-5-yl]formamido}-3-phenylpropanamide
3-benzyl-3-{2-[4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-1-methyl-2,3-dihydro-1H-indol-2-one
1-(4-{[3-(dimethylamino)butyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[2-(ethylsulfanyl)ethyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
1-cyclohexyl-3-(cyclopropylmethyl)-N-(oxan-4-ylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide