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2-(5-{2-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
N-{[6-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridin-3-yl]methyl}acetamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(1,3-thiazol-5-yl)propan-2-yl]benzamide
1-(2-{[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
2-(benzyloxy)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]ethan-1-one
N-cyclopentyl-2-({2-[(4-fluorophenyl)formamido]ethyl}amino)propanamide
N-methyl-N-[3-(oxolan-2-yl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(2-fluoro-4-methoxyphenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-phenyl-1H-pyrazole
7-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
1-(1-benzyl-1H-pyrazole-4-carbonyl)-4-(thian-4-yl)piperazine
ethyl 4-[(3-fluorophenyl)methyl]-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidine-4-carboxylate
3-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-3-carboxamide
N4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
[2-(1H-indol-3-yl)ethyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
2-[3-(3-phenylpropanoyl)piperidine-1-carbonyl]benzonitrile
5-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-{2-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]propan-1-one
1-({2-methoxy-5-[3-methyl-1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methyl)-1H-1,2,4-triazole
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(thiophen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-acetyl-8-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(2-hydroxybenzoyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-(1H-1,3-benzodiazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(1R,2S,9R)-11-(2-propylpyridine-4-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
3-(2-fluorophenyl)-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-pyrazole-5-carboxamide
1-(8-methyl-3-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)piperidine
2-amino-3-ethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-{[(1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)oxy]methyl}pyridine
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(3-methoxybenzoyl)piperidine
1-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(propylsulfanyl)ethan-1-one
2-[4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-1,3-benzoxazole
2-(2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
(1R,5R)-6-[(4-methanesulfonylphenyl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-6-methylpyridine-2-carboxamide
4-(4-chlorophenyl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)butanamide
2-(3-chloro-4-methoxyphenyl)-5-(methanesulfonylmethyl)pyridine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5,6-dimethylpyridine-3-carboxamide
3-{[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]sulfonyl}-N-propylbenzamide
1-(furan-2-ylmethyl)-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
4-cyclopentyl-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)pyrimidin-2-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
2-(5-acetylthiophen-3-yl)-1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]ethan-1-one
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(1,2-oxazol-3-ylmethyl)benzamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)thiophene-3-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
(2S,4S)-4-amino-1-methyl-N-[2-(N-methylmethanesulfonamido)ethyl]pyrrolidine-2-carboxamide
{4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]morpholin-2-yl}methanamine
4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one