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3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}propanamide
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[2-(methylsulfanyl)phenyl]urea
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethylbutan-1-one
N-[(5-methylpyrazin-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
3-[(3R,4S)-1-(4-chloro-2-hydroxybenzoyl)-4-(dimethylamino)piperidin-3-yl]propanoic acid
1-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(3-methyl-1-phenyl-1H-pyrazol-5-yl)urea
1-{5-[(2-methoxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
N-(4-{[methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenyl)acetamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-methyl-1H-pyrazole-5-carboxamide
N-(2-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}quinolin-6-yl)acetamide
7-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(3S,4R)-3-cyclopropaneamido-4-(4-methylphenyl)pyrrolidine-1-carbonyl]cyclopropane-1-carboxamide
2-{8-[(6-methylpyridin-2-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[2-(piperidin-1-yl)ethyl]acetamide
3-methyl-1-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-3-phenylpiperidine
2-methyl-7-[2-(propan-2-yl)pyrimidine-4-carbonyl]-2,7-diazaspiro[4.5]decane
5-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-2-(2-methoxyethyl)pyrimidine
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-methoxy-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydropyridin-2-one
2-(methoxymethyl)-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-benzoxazole
2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyridine
2-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperidin-3-yl)-1,3-benzoxazole
5-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
7-(cyclopropylmethyl)-2-[2-(4-fluorophenoxy)ethyl]-2,7-diazaspiro[4.5]decan-6-one
1-cyclopentyl-4-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-one
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-2-ethyl-N-(oxolan-2-ylmethyl)butanamide
(4aS,8aR)-6-(furan-2-ylmethyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
(4aS,8aS)-4a-hydroxy-N-[2-(piperidin-1-ylmethyl)phenyl]-decahydroisoquinoline-2-carboxamide
N-{2-[1-(9H-fluorene-9-carbonyl)piperidin-2-yl]ethyl}acetamide
2-(4-propanoylphenoxy)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
(1S,5R)-6-benzyl-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3-methylbutyl)-5-[4-(4-methylphenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-cyclooctyl-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-(cyclopropylmethyl)-8-(5-methylhexan-2-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-(2,4-dimethylphenyl)-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-6-[(4-methylphenyl)sulfanyl]pyrimidin-2-amine
2-cyclopropyl-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-1,3-benzoxazole-6-carboxamide
(2S,4R)-4-amino-1-(5-phenyl-1,2-oxazole-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
{1-[4-(3-cyclopentyl-1H-1,2,4-triazol-5-yl)phenyl]ethyl}dimethylamine
5-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)pyridine-2,4-diol
N-(oxan-4-ylmethyl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-ethyl-5-{1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,2,4-triazole
N-(cyclohexylmethyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
N-cyclobutyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
5-(2,5-dimethylbenzoyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-methyl-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-ol
2-(carbamoylamino)-N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
N2,N2-dimethyl-N4-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine