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2-[methyl({5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl})amino]ethan-1-ol
2-methyl-4-(4-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}phenyl)butan-2-ol
1-{4-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N,N,3-trimethyl-2-[(1-methyl-5-phenyl-1H-pyrazol-3-yl)formamido]butanamide
N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
1-(2-cyanobenzoyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)pent-4-enamide
1-(4-aminopyrimidin-2-yl)-4-(2H-1,3-benzodioxol-5-yloxy)piperidine-4-carboxylic acid
N-[(2-chlorophenyl)methyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(propan-2-yl)propanamide
2-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-{4-[(3,4-dichlorophenyl)methyl]piperazin-1-yl}pyridine-4-carboxamide
1-(dimethylamino)-3-(4-methoxy-2-{[4-(pyrimidin-4-yl)piperidin-1-yl]methyl}phenoxy)propan-2-ol
N-[(4-fluorophenyl)methyl]-2-(methylamino)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-benzylpiperidin-3-ol
N-methyl-4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}pyridin-2-amine
4-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2-dihydrophthalazin-1-one
methyl 5-{[4-(4-carbamoyl-1,3-thiazol-2-yl)piperazin-1-yl]methyl}-2-hydroxybenzoate
1-(furan-2-ylmethyl)-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}piperidine-3-carboxamide
2-(3-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}phenoxy)ethan-1-ol
1-(pyridin-4-yl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
N-methyl-3-oxo-N-phenyl-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-methyl-7-[2-(pyridin-2-yl)-1H-imidazol-1-yl]-1,2-dihydroquinolin-2-one
N-{1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]acetamide
1-(cyclopentylmethyl)-4-(3-methylpyridin-2-yl)piperazine
(3R,4S)-4-phenyl-1-(5-phenyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-amine
(2S,4R)-1-benzyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
5-(2,3-dichlorophenyl)pyridin-2-amine
1'-[(4-methanesulfonylphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2S,3S)-2-[(2-cyclopropyl-6-oxo-1,6-dihydropyrimidin-5-yl)formamido]-3-methylpentanamide
ethyl 5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
3-(cyclopropylsulfamoyl)-5-[4-fluoro-3-(hydroxymethyl)phenyl]benzoic acid
4-{[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}benzonitrile
1-(methoxymethyl)-N-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]cyclobutane-1-carboxamide
4,6-dimethyl-13-[(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)methyl]-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
3-(azepan-1-ylmethyl)-1-(cyclobutylmethyl)-3-hydroxypiperidin-2-one
N3-benzyl-N3-butyl-1-(cyclohexylmethyl)-N5,N5-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(2S)-1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
N-[(4-fluorophenyl)methyl]-N-methyl-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
7-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-hydroxy-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)pyrazine-2-carboxamide
3-cyclopropyl-5-(2-methyl-4-phenyl-1,3-thiazol-5-yl)-1H-1,2,4-triazole
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)acetamide
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylsulfanyl)ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-(cyclopentylsulfamoyl)-N-(furan-3-ylmethyl)benzamide
2-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1,3-benzothiazole-6-carboxamide