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N-benzyl[(1-benzylpiperidin-3-yl)amino]sulfonamide
5-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-2-(3-methylphenyl)pyrimidine
4-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}benzoic acid
5-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-2-(methoxymethyl)pyrimidine
1-{3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]butyl}-1H-pyrazole
N-{[2-(benzyloxy)phenyl]methyl}-2-(1-methylpiperidin-2-yl)acetamide
methyl 4-({2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamido}methyl)benzoate
1-(3-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-chloro-3-(2,4-dimethoxyphenyl)-1H-indazole
N2,N2,N4-trimethyl-N4-{[2-(methylamino)pyrimidin-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carbonyl)pyridin-1-ium-1-olate
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(3R,4R)-3,4-dimethyl-1-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]pyrrolidin-3-ol
(4aS,8aR)-6-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-pyrazol-1-yl)butan-1-one
5-{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-(4-{1-[1-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
N-{2-[1-(3-aminothiophene-2-carbonyl)piperidin-2-yl]ethyl}acetamide
(4aR,7aS)-1-benzyl-4-[(6-methylpyridin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[2-(3-acetylphenyl)-1H-imidazol-1-yl]-3-methoxybenzoic acid
N-methyl-6-[3-(5-methylfuran-2-yl)butyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-[2-(furan-2-ylmethoxy)phenyl]-4-(morpholin-4-yl)piperidine-1-carboxamide
3-[(3-phenyl-1H-pyrazol-4-yl)formamido]-N-(1,3-thiazol-2-yl)propanamide
5-cyclopropyl-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-oxazole-4-carboxamide
N3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N1,N1,N3-trimethylpiperidine-1,3-dicarboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(naphthalen-2-ylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 5-(6-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-(4-{[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}piperidin-1-yl)-2-methylpropan-1-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-(pyridin-3-yl)acetamide
1-amino-N-{2-[1-(2-methylpropyl)piperidin-3-yl]ethyl}cyclopentane-1-carboxamide
5,6-dimethyl-2-(4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-[2-(3,5-dimethoxyphenyl)ethyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4,5-dimethyl-6-(pyridin-4-yl)-2-(pyrrolidin-1-yl)pyrimidine
3-[2-(4-chlorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[1-(4-fluorophenyl)propyl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-4-methylpiperazine
methyl 2-[(3-{5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}phenyl)amino]acetate
ethyl 2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidine-1-carbonyl]amino}acetate
6-(4-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}piperazin-1-yl)pyrazine-2-carboxamide
4-(5-{2-[3-cyclopropyl-1-(4-methylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
(1S,3R)-3-amino-N-{3-[methyl(phenyl)amino]propyl}cyclopentane-1-carboxamide
N-[3,3-dimethyl-1-(pyrrolidin-1-yl)butan-2-yl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
N-[2-(4-chlorobenzenesulfonamido)ethyl]-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-{4-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
(2R,3R,6R)-5-(1H-indole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{3-methyl-1-oxo-1-[4-(pyrimidin-2-yl)piperazin-1-yl]pentan-2-yl}-2,3-dihydro-1H-isoindol-1-one
(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
(4S)-3-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-4-phenyl-1,3-oxazolidin-2-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1,4-diazepane