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N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{1-cyclopentyl-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]benzoate
N-(3-acetylphenyl)-3-(2-{[(2-fluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carboxamide
(3R,4R)-4-(hydroxymethyl)-1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-ol
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)({[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl})methylamine
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-methyl-1H-1,3-benzodiazole-4-carboxamide
1-tert-butyl-4-({[(6-chloroquinolin-2-yl)methyl](methyl)amino}methyl)pyrrolidin-2-one
2-[(2-propoxypropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(prop-2-en-1-yl)(pyridin-2-ylmethyl)(quinolin-4-ylmethyl)amine
2-[(2-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]carbamoyl}phenyl)amino]acetic acid
2-methoxy-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
3-{1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
3-[methyl({2-methylthieno[2,3-d]pyrimidin-4-yl})amino]propane-1,2-diol
2-{1-[(3,4-difluorophenyl)methyl]-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
methyl 3-[3-(4-methylphenyl)propanoyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(1,4-dioxan-2-ylmethyl)-3-methoxybenzamide
(furan-2-ylmethyl)(3-methylbutan-2-yl)(quinoxalin-2-ylmethyl)amine
N-(3-ethoxypropyl)-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
3-(2-oxoazepan-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
2-ethyl-4-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}pyrimidine
1-{3-[2-(2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]morpholin-4-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-fluoro-6-methoxybenzamide
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-[3-(trifluoromethyl)phenyl]acetamide
5-[1-(3-chloro-4-ethoxybenzoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
N-{2-[4-(1H-indol-2-ylmethyl)morpholin-2-yl]ethyl}methanesulfonamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[(3-methylpiperidin-3-yl)methoxy]pyridine-3-carboxamide
ethyl 1-ethyl-5-[2-(1H-imidazol-2-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(4-acetylphenyl)-3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carboxamide
1-[3-(3-ethylphenoxy)propyl]-1-methyl-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)(4,4,4-trifluorobutyl)amine
1-(2-aminoethyl)-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1H-1,2,3-triazole-4-carboxamide
(2E)-1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-methylbut-2-en-1-one
methyl 2-[3-(4-chlorophenyl)-N-methyl-3-phenylpropanamido]acetate
4-{4-[3-(4-chlorobenzoyl)piperidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
7-(2-methoxyphenyl)-2-(propoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-methyl-2-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
(2S)-2-({1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-4-methylpentanamide
N-[(3S,4R)-1-(3-cyano-2-methoxypyridin-4-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
4-chloro-2-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-6-phenyl-N-propyl-1,2-dihydropyridine-3-carboxamide
[(3,4-difluorophenyl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-ethyl-4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
1-{4-[1-(furan-2-ylmethyl)piperidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-(6-methoxy-2H-1,3-benzodioxol-5-yl)urea
propan-2-yl 2-chloro-5-(5-propyl-1,2-oxazole-3-amido)benzoate
3-{[(4-chlorophenyl)methyl]amino}-N-(3-fluorophenyl)propanamide
(2S)-2-amino-4-hydroxy-1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
2-(4-methylphenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]quinoline-4-carboxamide