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3-cyclobutyl-4-[(1s,4s)-4-aminocyclohexyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(1-{[1-(2,4-dimethylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
5-(3-acetylphenoxymethyl)-N-(2-hydroxybutyl)-1,2-oxazole-3-carboxamide
6-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]pyrimidin-4-ol
N-(2-methoxyethyl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(propan-2-yl)acetamide
(3R,5S)-N-(4-fluorophenyl)-5-(piperidine-1-carbonyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N-(2-chloro-4,6-dimethylphenyl)-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
N,5,7-trimethyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
(4aS,7aR)-1-[2-(azocan-1-yl)acetyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-4,6-dioxo-3-[2-(propylsulfanyl)pyrimidin-5-yl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-(1H-1,2,3,4-tetrazol-5-yloxy)aniline
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[2-(pyridin-2-yl)acetyl]pyrrolidine-2-carboxamide
3-acetamido-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
1,5-dimethyl-2-phenyl-4-{[4-(4,6,7-trimethylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
3-[5-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(1-hydroxycyclopentyl)ethyl]amino}methyl)piperidin-2-one
1-[2-(3-fluorophenyl)ethyl]-N-[2-(1H-indol-3-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl (2S,4S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]propanamide
1-methyl-1-{3-[(4-methylphenyl)sulfanyl]propyl}-3-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}acetamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-2-ynamide
4-acetyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)benzamide
methyl 2-[benzyl(methyl)sulfamoyl]-6-butanoyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
7-[2-(3-chloro-4-hydroxyphenyl)acetyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide
butyl 4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxylate
1-(2-{[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
4-{[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
N3-cyclooctyl-N5-(3-ethoxypropyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(1-propylpiperidin-4-yl)-2,3-dihydro-1H-indene-2-carboxamide
(2S,4S)-4-[3-(trimethyl-1H-pyrazol-4-yl)propanamido]pyrrolidine-2-carboxylic acid
1-[(4-methanesulfonylphenyl)methyl]-2-(3-methoxyphenyl)piperidine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-methylpyrimidine-5-carboxamide
5-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)morpholine
2-(2-{4-phenyl-1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-5-yl}-1H-pyrrol-1-yl)pyridine
methyl 2-({4-[(pyrimidin-2-yl)amino]piperidin-1-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
2-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-4-[(1-methyl-1H-pyrrol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-2,2-dimethylmorpholine
ethyl 5-(1-benzyl-1H-pyrazole-4-carbonyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)propanamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[3-(1H-imidazol-2-yl)propyl]urea
7-chloro-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine