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N-(1,2-oxazol-3-ylmethyl)-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamide
4-[4-(morpholine-4-carbonyl)benzenesulfonyl]-1,4-oxazepane
6-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine-2,4-diamine
N4-[(1R,3R)-3-aminocyclopentyl]-6-[(4-fluorophenyl)sulfanyl]pyrimidine-2,4-diamine
N-(1-benzylpyrrolidin-3-yl)-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
2-(3,4-dimethoxyphenyl)-N-(oxolan-3-yl)acetamide
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-N,N-diethylacetamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-phenoxypropanamide
3-{[(adamantan-2-yl)amino]methyl}-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-(pyridin-4-yl)propanamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
5-(methoxymethyl)-N-[(4-phenyloxan-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-propylpyridine-4-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-[2-(2-methoxyethoxy)phenyl]-3-[1-(oxan-4-yl)piperidin-4-yl]urea
7-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
methyl 5-{[(2-fluorophenyl)methyl]amino}-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(1H-indol-3-yl)-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,2-dimethyl-1-benzofuran-5-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
ethyl 1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-imidazole-2-carboxylate
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-4-(piperidin-1-ylmethyl)benzamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,3-dimethyl-1H-indole
2-[(4-fluorophenyl)methyl]-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}morpholine
N-[2-(2,5-dimethylphenoxy)ethyl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
1-{4-[(2-ethoxypropyl)(methyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-{1-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
4-(3-{[1-(oxolane-3-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
7,7-dimethyl-2-(morpholin-4-yl)-N-(quinolin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
(3S,4S)-4-[(2-amino-5-methylpyrimidin-4-yl)amino]-1-(propan-2-yl)pyrrolidin-3-ol
3-[1-methyl-5-(3,4,5-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
N-[4-chloro-3-({[3-(1H-1,2,3-triazol-1-yl)propyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(3-methoxypropyl)-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine-3-carboxylic acid
4-methyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pentanamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-cyclobutanecarbonyl-4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-2-amine
8-[(2-ethylphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(3S)-3-hydroxy-3-phenylpropyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
8-chloro-2-({[1-(3,4-dimethoxyphenyl)ethyl]amino}methyl)quinolin-4-ol
2-[(furan-2-ylmethyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amino]butan-1-ol
3-methyl-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1-(2-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-chloro-N-(2-methoxyethyl)-4-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]oxy}benzamide
(2S,4R)-4-amino-1-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-N-ethylpyrrolidine-2-carboxamide