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N-[(3S,4R)-1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-propyl-4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}pyrrolidin-2-one
8-(isoquinolin-5-yl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-{3-[(dimethylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-{4-[2-(tert-butylsulfamoyl)phenyl]phenyl}-N-methylacetamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2,2,2-trifluoroethyl)benzamide
N-(2-fluoro-5-methylphenyl)-4-oxo-4-[4-(1,3,5-triazin-2-yl)piperazin-1-yl]butanamide
3-(prop-2-en-1-yl)-1-(4-sulfamoylbutanoyl)piperidine-3-carboxylic acid
1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
(2-{5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-3-methyl-1H-pyrazol-1-yl}ethyl)dimethylamine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-decahydro-1,6-naphthyridin-2-one
N-[2-(dimethylamino)ethyl]-3-({1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}propanamide
8-benzyl-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-hydroxy-7-methoxy-4-(2-phenylphenyl)-1,2,3,4-tetrahydroquinolin-2-one
(1R,5S,8R)-3-[(6-fluoroquinolin-2-yl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
5-(3,4-difluorophenoxymethyl)-N-(oxolan-3-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
2-(4-methanesulfonylphenyl)-6-(pyrrolidine-1-carbonyl)pyrazine
N-methyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]benzamide
N3-(cyclohexylmethyl)-N5-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-{5-[({[(2R,3R,5S)-2-(4-chlorophenyl)-1-ethyl-5-(hydroxymethyl)-5-methylpyrrolidin-3-yl]methyl}amino)methyl]thiophen-3-yl}prop-2-yn-1-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-methylpyrimidin-5-yl)methyl]piperidin-3-ol
8-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-1-oxa-8-azaspiro[4.5]decane
5-methyl-1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-5-phenylpiperidin-2-one
N-cycloheptyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide
[1-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)piperidin-3-yl]methanol
1'-(cyclohexylmethyl)-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}azepane-2-carboxamide
5-[2-(4-fluorophenoxy)ethyl]pyridine-3-carboxamide
2-(2-methyloxane-2-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(1-methyl-1H-indol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)urea
2-methyl-5-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyrazine
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)cyclopropan-1-amine
3-(4-chlorobenzoyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidine
N-cyclopropyl-1-{4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanoyl}piperazine-2-carboxamide
1-[2-(1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
2-{[(dimethyl-1,3-thiazol-5-yl)methyl]amino}-N-[(4-acetamidophenyl)methyl]acetamide
N-[2-(dimethylamino)ethyl]-4-{furo[3,2-c]pyridin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-methyl-1-benzofuran-5-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)(1,4-dioxan-2-ylmethyl)methylamine
2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1H-imidazole
N-[2-(methylsulfanyl)phenyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
(2R,4S)-1-[(2-carboxyphenyl)methyl]-4-hydroxypiperidine-2-carboxylic acid
2-(4-{[2-(pyrrolidin-1-yl)ethyl]amino}piperidin-1-yl)pyridine-4-carbonitrile