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5-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(propan-2-yl)pyridine-3-carboxamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
N-methyl-N-{2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}methanesulfonamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
5-cyclopropanecarbonyl-1'-(1H-1,2,4-triazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(5-fluoro-2-methoxybenzoyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-1-one
(1S,5R)-6-[(2-phenylpyrimidin-5-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(1-ethylpiperidin-4-yl)ethyl]-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-5-fluoro-N-methylpyrimidin-4-amine
2-phenyl-4-{1-[3-(1H-pyrazol-1-yl)propyl]-1H-imidazol-2-yl}-1,3-oxazole
1-(5-chlorothiophene-2-carbonyl)-4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine
3-[(2R,3R,6R)-5-(5-methyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-{2-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
4-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]benzoic acid
4-[2-(3-fluoro-4-methylphenyl)acetyl]piperazine-2-carboxylic acid
N-[2-methoxy-5-({methyl[1-(3-methylpyridin-2-yl)propan-2-yl]carbamoyl}amino)phenyl]propanamide
3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
1,3-dimethyl-5-{2-oxo-2-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}imidazolidine-2,4-dione
N-{4-[(methylcarbamoyl)methyl]phenyl}-4-(oxan-4-yl)piperazine-1-carboxamide
3-({1-[4-(1H-pyrazol-1-yl)butanoyl]pyrrolidin-3-yl}methyl)benzoic acid
4-(2-fluorophenoxy)-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxylic acid
1,3,6-trimethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-benzyl-3-(piperidin-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(dimethylamino)-N-ethyl-2-(4-fluorophenyl)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-[(3S,4R)-4-(4-methylphenyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]acetamide
5-[1-(difluoromethyl)-3-methyl-1H-pyrazol-4-yl]quinoline
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)urea
{1-[7-chloro-2-(furan-2-yl)-8-methylquinoline-4-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
2-(pyridin-2-ylmethyl)-8-(1,3-thiazol-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]propan-1-one
N-{4-[(2S)-2-acetamido-3-(1H-imidazol-4-yl)propanamido]phenyl}pentanamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(quinoline-2-carbonyl)pyrrolidin-3-yl]methanol
5-[(1S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1,3-benzoxazole
1-{4-[3-(4-fluorophenoxy)azetidine-1-carbonyl]phenyl}piperidine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(morpholin-4-yl)propan-1-one
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
7-chloro-3-[(3-propoxypiperidin-1-yl)methyl]-1,2-dihydroquinolin-2-one
4-(4-methanesulfonylphenyl)-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[4-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-[2-(aminomethyl)morpholine-4-carbonyl]-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
N-{4-[(2-benzylmorpholin-4-yl)methyl]phenyl}acetamide
1-[1-(ethanesulfonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-8-fluoro-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-methyl-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
methyl (2S)-1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
methyl 2-[(2-methylphenyl)sulfamoyl]-6-(4,4,4-trifluorobutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}piperidine-1-carboxylate