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ethyl 3-[(2-methylphenyl)methyl]-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine-3-carboxylate
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]acetamide
methyl 4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}benzoate
5-(2,4-difluorophenoxymethyl)-N-[1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
2-(2-aminoethyl)-N-ethyl-N-[(1-ethylpyrrolidin-3-yl)methyl]quinazolin-4-amine
1-[(4-hydroxy-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}azepan-4-yl)methyl]-3,3-dimethylurea
4-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}-1,4-oxazepan-6-ol
4-[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]-6-(methoxymethyl)pyrimidine
N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-2-phenylbutanamide
3,8-bis(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N3-(1,3-benzothiazol-2-ylmethyl)-N5-benzyl-1-cyclopropyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
(2S)-2-(1,2-oxazol-3-ylformamido)-3-phenylpropanamide
(diphenylmethyl)({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
1-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-methoxy-5-{1-[(3S,4R)-4-methoxyoxolan-3-yl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
(4aS,8aR)-6-(5-chloropyridin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(2E)-1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-phenylprop-2-en-1-one
2-(4-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-cyclopentyl-1,5-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrazole-3-carboxamide
8-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(1,4-dioxan-2-ylmethyl)(methyl){[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(quinolin-6-ylmethyl)propanamide
N-cyclooctyl-2-{methyl[(1-methylpyrrolidin-2-yl)methyl]amino}acetamide
N-ethyl-2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
2-(2,3-dimethylphenoxy)-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]acetamide
3-chloro-N-cyclopentyl-4-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}oxy)benzamide
4-(1H-imidazol-1-yl)-1-[5-(propan-2-yl)thiophene-3-carbonyl]piperidine-4-carboxylic acid
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
3-fluoro-N-{1-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
6-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-benzyl-2-{[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
1-(2-aminoethyl)-N-butyl-N-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-phenoxypiperidine-4-carboxylic acid
{2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-8-methylquinolin-3-yl}methanol
1-cyclopentyl-4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-2-one
1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]-3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyrimidin-4-amine
[(4-fluorophenyl)methyl]({[3-(1H-pyrazol-1-yl)phenyl]methyl})(pyridin-4-ylmethyl)amine
3-phenyl-4-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)-1H-pyrazole
1-(cyclohexylmethyl)-5-(4-ethylpiperazin-1-yl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyridine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methylimidazo[1,2-a]pyridine-6-carboxamide
1-cyclopropanecarbonyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]piperidine-4-carboxamide
(3R,5S)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1-methyl-1H-pyrazole-3-carboxamide
2-(methoxymethyl)-1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
(4aS,8aR)-6-(2,5-dimethylfuran-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one