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N-{[5-(methoxymethyl)furan-2-yl]methyl}-4-methyl-5-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(methylsulfanyl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
1-(oxan-4-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine-3-carboxamide
4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]-N-[(1R)-1-(4-methoxyphenyl)ethyl]piperidine-1-carboxamide
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(4-methylpyridin-2-yl)methyl]benzamide
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-(pyridin-2-yl)pyrimidin-2-amine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-methoxy-N-methylbenzamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propan-1-one
3-[1-({5-[1-(3-fluoropropyl)-1H-pyrazol-3-yl]furan-2-yl}methyl)pyrrolidin-2-yl]-4-methyl-1,2,5-oxadiazole
N-ethyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
2-(4-{[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]methyl}phenyl)acetic acid
1-[(5-ethylpyridin-2-yl)methyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-methylurea
1-(2-methoxyphenyl)-4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[4-(1H-pyrazol-1-yl)butan-2-yl]amine
2-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-N-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
ethyl 4-{4-[(2-fluorophenyl)methyl]-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl}piperazine-1-carboxylate
N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]amino}acetamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(3R,4S)-4-cyclopropyl-1-(furan-2-ylmethyl)pyrrolidin-3-amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylfuran-3-carboxamide
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
2-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-cyclopentyl-N3-(3-methylbutyl)-4-oxo-N5-[2-(pyrrolidin-1-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(3-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrazine
8-[(4-methoxyphenyl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S)-3-benzyl-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-2-one
4-(2-ethylpyrimidine-5-carbonyl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-cyclopropyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
3-(4-ethyl-1H-pyrazol-5-yl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
8-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}propan-1-one
5-(2-methoxyphenoxymethyl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[1-(4-ethoxyphenyl)ethyl]-N-methyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
{2-[2-(2-ethyl-1-benzofuran-3-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
N-methyl-N-(pyrazin-2-ylmethyl)-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
[(1-cyclopentylpiperidin-4-yl)methyl][(4,5-dimethylfuran-2-yl)methyl](pyridin-3-ylmethyl)amine
2-(3-methoxypropyl)-8-[(4-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(2-methoxyacetyl)-N-methylpiperidine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl]methanesulfonamide
N-[2-(3-methoxyphenyl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{3-[4-(4-chlorophenyl)-4-hydroxypiperidine-1-carbonyl]piperidin-1-yl}-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
7-[2-(ethylamino)pyrimidine-5-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-(2-methoxyacetyl)-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-fluoropyridin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one