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4-(4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
3-{[2-(3-methoxypropyl)piperidin-1-yl]sulfonyl}pyridine
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-[(4-methylphenyl)sulfanyl]propanamide
3-[4-(1H-pyrazol-5-yl)phenyl]-1-[(1r,4r)-4-hydroxycyclohexyl]urea
N-[(3S)-1-[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl]acetamide
8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(1S,6R)-9-(1H-1,3-benzodiazole-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4-methyl-1,3-benzothiazol-2-amine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(3-fluorophenyl)-2-hydroxyethyl]benzamide
5-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-4-phenylpyrimidin-2-amine
3-(4-methoxy-3,5-dimethylbenzoyl)-1-(1,2,3-thiadiazole-4-carbonyl)piperidine
1-tert-butyl-5-oxo-N-[2-(1,3-thiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
1-[(2S)-oxolan-2-ylmethyl]-5,5-diphenylpiperidin-2-one
1-[6-methyl-2-(methylamino)pyrimidin-4-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N,N-dimethyl-5-{[(oxan-4-yl)carbamoyl]amino}-1-benzothiophene-2-carboxamide
4-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3,5-trimethyl-1H-pyrazole
4-(benzyloxy)-1-(oxolane-3-carbonyl)piperidine
N-(4-acetylphenyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
2-(3-fluoro-4-hydroxyphenyl)-1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
4-(5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
(2S)-N-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-2-(methoxymethyl)pyrrolidine-1-carboxamide
3-benzyl-1-(3-methoxypropyl)-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-methyl-1H-pyrrole-2-carbonyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-{3-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]propoxy}benzamide
1-[(4-ethylphenyl)methyl]-5-[5-(methoxymethyl)furan-2-yl]-1H-1,2,4-triazole
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(2-methylpropyl)-8-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
2-{2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
3-{2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-4-(3-methylbut-2-en-1-yl)piperazin-2-one
11-(pyrrolidin-3-yl)-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-12-one
2-[3-(2-phenylethyl)-5-[2-(1H-1,2,4-triazol-5-yl)phenyl]-1H-1,2,4-triazol-1-yl]pyridine
(2S,4S)-N-ethyl-4-(3-methoxypropanamido)-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-2-carboxamide
2-(3-fluoro-4-hydroxyphenyl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)acetamide
(4aS,8aR)-1-(2-aminoethyl)-6-(5-methyl-1-benzofuran-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
(1S,5R)-6-[(5-chlorothiophen-2-yl)methyl]-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
ethyl (2S)-2-{[1-(2-fluorophenyl)cyclopropyl]formamido}propanoate
7-(3-chlorophenyl)-4-(2-hydroxybenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-methyl-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}thiophene-2-sulfonamide
2-(2-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}phenoxy)acetic acid
(4S)-3,3,4-trimethyl-1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidin-4-ol
(3S,4S)-1-(benzenesulfonyl)-4-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]pyrrolidin-3-ol
1-methyl-4-[(4-methyl-5-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]piperazine
6-methyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
N-(2-methyl-1-oxo-1-{2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}propan-2-yl)thiophene-2-carboxamide
2-[1-(2-hydroxyethyl)-5-(5-methyl-4-phenylthiophen-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
5-ethanesulfonamido-1-methyl-N-[2-(methylsulfanyl)ethyl]-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1,4-diazepan-1-yl}-4,6,7-trimethylquinazoline