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3-[5-(piperidin-1-ylmethyl)pyridin-2-yl]aniline
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2-fluorophenyl)methyl]pyrrolidine-2-carboxylate
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
4-chloro-3-methyl-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-5-carboxamide
(1S,5R)-6-[(2,3-dimethoxyphenyl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(2-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]-1-methylpiperazin-2-one
2-(3-methyl-5-{[(1-methyl-1H-indol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl)acetic acid
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methylfuran-2-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine-3-carboxylate
2-(2-chloro-4-fluorophenoxymethyl)-4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazole
2-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2,3-dihydro-1H-isoindole
5-cyclopropyl-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-(naphthalen-1-ylmethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
1-{3-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}-1H-pyrazole
5-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-3-(2-methylpropyl)-1,2-oxazole
4-(1-benzofuran-2-carbonyl)-2-[(3-methoxyphenyl)methyl]morpholine
5-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-6-methylquinoline
2-(2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-oxoethyl)cyclopentan-1-one
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-[2-(thiophen-3-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-(2-methoxyphenyl)-N-(oxan-4-ylmethyl)pyridazin-3-amine
2-amino-4-(2-butyl-1H-imidazol-4-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
diethyl({3-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
N-(1-carbamoylcyclopentyl)-7-chloro-3,5-dimethyl-1-benzofuran-2-carboxamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2H-1,3-benzodioxole-5-carboxamide
1-(cyclopropylmethyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-phenyl-1-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-4-carbonitrile
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(5-methylthiophen-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
7-cyclopentyl-2-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(2R,5R)-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2,5-dimethyl-4-(prop-2-en-1-yl)piperazine-1-carboxamide
(3S,4S)-4-cyclopropyl-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidine-3-carboxylic acid
4-(5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
2-{[(3R,4S)-1-(2-methoxyacetyl)-4-propylpyrrolidin-3-yl]amino}-5,6-dimethylpyridine-3-carboxamide
2-[1-(2,4-dimethylphenyl)-5-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
7-(2,2-dimethylpropyl)-2-[2-(phenylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-amino-2-methyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
4-(2,6-dimethoxyphenyl)-2-methyl-1H-imidazole
1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-7-(3-methoxypropanamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
2-(9-{[2-(2-hydroxyethoxy)phenyl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetamide
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-4-(pyridin-4-yl)pyrimidin-2-amine
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-(6-methoxypyridin-3-yl)-1-methylpyrrolidine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-3-(2-methylphenyl)propanamide
2,3-difluoro-4-methoxy-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)benzamide
1,3-dimethyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
[(2S)-1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-2-yl]methanol