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N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-[1-(2,4-dimethoxyphenyl)ethyl]-1-[2-(ethylsulfanyl)phenyl]-3-methylurea
3-(1H-1,3-benzodiazol-2-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
3-chloro-5-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
6-[3-(2,4-dichlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
2-[8-(1H-indol-3-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
5-[(3-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(3-methoxyphenyl)-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}propanamide
(4aS,7aR)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[5-cyclopropyl-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-(4-methoxyphenoxy)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
6-(1-methylpiperidin-3-yl)-2-[2-(trifluoromethyl)phenyl]-3,4-dihydropyrimidin-4-one
3-(5-methyl-1H-pyrazol-1-yl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]propanamide
(2R,6R)-4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(5-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
3-[(cyclohexylmethyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
(3S,4S)-4-cyclopropyl-1-[2-(3-fluorophenyl)acetyl]pyrrolidine-3-carboxylic acid
8-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-methyl-3-{[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(2-methoxyethyl)-2-(pyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(3aR,6aS)-5-(2,1-benzoxazole-3-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-(3-chlorobenzoyl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(prop-2-en-1-yl)amine
N-cyclohexyl-2-cyclopropyl-6-oxo-N-(pyridin-2-ylmethyl)-1,6-dihydropyrimidine-5-carboxamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
2-(3-{5-[5-(hydroxymethyl)furan-2-yl]-4-phenyl-1H-imidazol-1-yl}propyl)phenol
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-5-methylpyrazine-2-carboxamide
3-{[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]methyl}benzonitrile
5-[(4,5-dimethylfuran-2-yl)methyl]-3-[(phenylsulfanyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-methyl-6-oxo-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,6-dihydropyridine-3-carboxamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[4-(1H-pyrazol-1-yl)butan-2-yl]benzamide
1-benzoyl-4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazine
N-cyclohexyl-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(prop-2-yn-1-yl)benzamide
1-cyclohexyl-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-amino-4-(1H-imidazol-4-yl)-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(3R,5S)-5-[3-(dimethylamino)pyrrolidine-1-carbonyl]-N-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
2-{1-[(3-chlorophenyl)methyl]pyrrolidin-2-yl}pyridine
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-[2-(dimethylamino)ethyl]-9-[(4-methoxy-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-hydroxy-3-{[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-(2-phenylethyl)piperidin-2-one
1-{3-[(1-benzofuran-2-ylmethyl)amino]-5-(dimethylsulfamoyl)benzoyl}piperidine-3-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
2-{3-[3-(4-methylpyridin-3-yl)phenyl]-1H-pyrazol-1-yl}-N-(pyrazin-2-yl)acetamide
2-[5-(4-chloro-3-methyl-1H-pyrazol-5-yl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
1-[3-({7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenyl]ethan-1-one
4-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one