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6-[4-(3-fluorophenoxy)piperidin-1-yl]pyridine-3-carboxylic acid
methyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})(1H-pyrazol-5-ylmethyl)amine
1-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
benzyl(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
4,5-dimethyl-2-{2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,3-benzodiazole
2-(1-cyclohexyl-4-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
{4-[({2-cyclopentyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}(methyl)amino)methyl]oxan-4-yl}methanol
3-(1-{[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-1-ol
5-(2-methylpropyl)-1'-(6-methylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 1-{7-methylpyrazolo[1,5-a]pyrimidine-6-amido}piperidine-3-carboxylate
1-(1-methyl-5-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}-1H-pyrrol-3-yl)ethan-1-one
4-(4-cyclopropanecarbonylpiperazin-1-yl)-2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(3S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
4-[3-(piperidin-4-ylmethyl)benzoyl]-3-propylmorpholine
2-(1-benzoxepine-4-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(carbamoylamino)acetamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-methoxy-N-methyl-4-oxo-1,4-dihydropyridine-2-carboxamide
4-(3-chlorophenyl)-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-amido}oxane-4-carboxylic acid
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[4-(pyrrolidin-1-yl)benzoyl]piperidine
N-{1-[(3-methylphenyl)methyl]cyclopropyl}oxane-2-carboxamide
methyl (2R,4S)-4-hydroxy-1-(3-methylbut-2-en-1-yl)piperidine-2-carboxylate
2-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-[5-(4-acetylphenyl)-4-phenyl-1H-imidazol-1-yl]-N-methylbutanamide
1-[4-(3-methoxyphenyl)phenyl]-N-(pyridin-4-ylmethyl)piperidin-4-amine
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2,3-dimethyl-1H-indole-7-carboxamide
[(3R,4R)-1-[(4-chloro-2-fluorophenyl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
4-phenyl-3-(piperidin-4-yl)-1-[3-(1H-pyrrol-1-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 2-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
(1R,5S,6R,7S)-3-(2-aminoethyl)-6-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]decan-4-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
5-[3-(2-methoxyphenyl)-1H-pyrazol-5-yl]-3-methyl-1H-1,2,4-triazole
N-[(3S,4R)-4-(4-methylphenyl)-1-(oxane-4-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide
(2S,4S)-4-amino-1-[2-(2,5-dimethylphenyl)acetyl]-N-ethylpyrrolidine-2-carboxamide
1-(2-chloro-3-methoxyphenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methylurea
N5-[3-(morpholin-4-yl)propyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-[(1S,5R)-3-(2-chloro-4-fluorobenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-{1-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]piperidin-4-yl}-N-methylacetamide
(3R,4R)-1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-4-(hydroxymethyl)piperidin-3-ol
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-4-(1H-imidazol-2-yl)piperidine
2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-5-propyl-1,3,4-oxadiazole
1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-(1H-indol-2-ylmethyl)-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(6-hydroxy-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one