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5-fluoro-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1,3-dimethyl-1H-indole-2-carboxamide
3-(4-hydroxyphenyl)-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-5-carboxamide
3-ethyl-8-{spiro[2.3]hexane-1-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-({3-[(2S)-4-methyl-2-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
1-(furan-2-carbonyl)-4-(2-methyl-4-phenylpyridine-3-carbonyl)-1,4-diazepane
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-3-(methoxymethyl)pyrrolidine-1-carboxamide
3-(piperidin-1-ylmethyl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-ol
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)benzamide
4-(2-hydroxyethyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[2-(propan-2-yloxy)-5-({[1-(pyrimidin-2-yl)piperidin-3-yl]amino}methyl)phenyl]methanol
(3aR,6aR)-2-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(4aR,7aS)-1-(2-phenylethyl)-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,4S)-5-[(2,6-difluorophenyl)methyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(pyridin-3-ylmethyl)-9-(pyridine-3-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
1-(4-cyanonaphthalen-1-yl)-3-[2-(1-hydroxycyclopentyl)ethyl]-3-methylurea
{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
2-butoxy-N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}acetamide
1-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]-3,5-dimethyl-1H-pyrazole
(3E)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)hex-3-enamide
N,N-dimethyl-3-[1-methyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]aniline
N-[(2-fluorophenyl)methyl]-2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]acetamide
4-[(6-methylpyridin-3-yl)oxy]-N-(oxan-2-ylmethyl)piperidine-4-carboxamide
4-{[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl](methyl)amino}-N-(furan-3-ylmethyl)pyridine-2-carboxamide
(3R,4R)-1-(4-ethyl-5-methylpyrimidin-2-yl)-3,4-dimethylpyrrolidin-3-ol
(1S,6R)-3-(5-fluoro-2-methoxybenzoyl)-3,9-diazabicyclo[4.2.1]nonane
1-(3-chlorophenyl)-3-(oxan-4-yl)-5-{pyrazolo[1,5-a]pyrimidin-2-yl}-1H-1,2,4-triazole
N,N-dimethyl-2-[(thiophen-2-ylformamido)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
2-[3-(2-methoxyethyl)-5-[2-(3-methylphenoxy)propan-2-yl]-1H-1,2,4-triazol-1-yl]acetic acid
2-amino-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[cyclopropyl(pyridin-2-yl)methyl]-N,2-dimethyl-3-[(pyridin-3-ylmethyl)amino]benzamide
1-(diphenylmethyl)-N-(3-hydroxy-3-phenylpropyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
N,8-dimethyl-N-(2-phenylethyl)-3-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
3-chloro-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyridine-4-carboxamide
3-[1-(2,3,4-trifluorophenyl)-1H-imidazol-2-yl]benzonitrile
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(piperidin-1-yl)ethyl]acetamide
[(5-cyclopentylthiophen-2-yl)methyl](ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
1-cyclohexyl-4-[6-(thiomorpholin-4-yl)pyridine-3-carbonyl]-1,4-diazepane
(1S,5R)-6-propyl-3-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[(2S)-2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidin-1-yl]ethan-1-one
1-(5-propyl-1,2-oxazole-3-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
3-chloro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-propoxybenzamide
5-(4-aminoazepane-1-carbonyl)-N-(2-methoxyethyl)-1-methyl-1H-1,3-benzodiazol-2-amine
(3aR,6aR)-2-[2-(2-ethylphenoxy)ethyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[3-(trifluoromethyl)phenyl]-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazole
3-[(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide