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N-(3-fluorophenyl)-1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
N-ethyl-6,6-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-oxothiomorpholine-3-carboxamide
1-[2-({4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)morpholin-4-yl]ethan-1-one
2-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}pyridine-4-carboxamide
(2S,4R)-1-[(4-chlorophenyl)methyl]-N,N-diethyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}butan-1-one
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,5-dimethoxybenzamide
2-[4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazin-1-yl]ethan-1-ol
3-[3-(cyclopentylcarbamoyl)propanamido]propanoic acid
2-(4-{[4-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
N-({1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}methyl)cyclopropanecarboxamide
5-(furan-2-ylmethyl)-5-{3-oxo-3-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propyl}pyrrolidin-2-one
4-(1H-1,3-benzodiazol-1-yl)-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine-4-carboxylic acid
1-({5-[(5-hydroxy-2-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
7-chloro-2-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]quinoxaline
4-({2-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-2-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]quinoline
(2R)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}oxolane-2-carboxamide
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-(4-methylphenoxy)ethan-1-one
4-(4-chlorophenyl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}butanamide
4,4-difluoro-N-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)piperidine-1-carboxamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
methyl 5-({[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}amino)-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-(trifluoromethyl)morpholine
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-tert-butyl-3-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1H-pyrazole
4-(2-benzyl-3-oxopiperazine-1-carbonyl)-N,N-dimethylpiperidine-1-carboxamide
6-{[methyl({[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl})amino]methyl}-1,4-oxazepan-6-ol
2-{[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](thiophen-3-ylmethyl)amino}butan-1-ol
N-[2-(2-ethoxyphenyl)ethyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-(3-cyclopentylpropyl)-N-methyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
4-methyl-6-(propan-2-yl)-2-{4-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-1-yl}quinazoline
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[2-(2-methoxyphenyl)ethyl]pyrrolidine-2-carboxamide
3-(4-fluorophenyl)-4-(2,3,4-trimethoxybenzoyl)piperazin-2-one
2-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
(1R,3S,5S)-8-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
4-(2,4-difluorophenyl)-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-6-methylpyridine-3-carboxylic acid
[(3R,4R)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-[3-({[(2-fluorophenyl)methyl](2-hydroxyethyl)amino}methyl)phenyl]-5,6-dimethyl-3,4-dihydropyrimidin-4-one
3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methyl-1-[4-(1H-pyrazol-5-yl)phenyl]urea
2-(cyclopropylmethyl)-8-(8-methoxyquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-(4-{[2-(2,5-dimethylphenoxy)ethyl](methyl)amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[2-(dimethylamino)ethyl]-3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]propanamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
5-{5-[(2S)-butan-2-yl]-1,2,4-oxadiazol-3-yl}-6-methyl-2-(4-methyl-1H-imidazole-2-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2-methyl-N-(oxolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(3R,4R)-1-[3-(dimethylsulfamoyl)propyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide