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(2S)-2-amino-4-hydroxy-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
N-[4-({7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)phenyl]acetamide
1-[1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
5-{5-[1-(propan-2-yl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
2-{1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-N-[(2-methoxyphenyl)methyl]acetamide
ethyl 3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2,6-dimethyl-8-[(1-phenylpiperidin-4-yl)amino]octan-2-ol
N,N-dimethyl-4-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)piperazine-1-carboxamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-(2-oxopiperidin-1-yl)acetamide
N-[1-(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methylpropyl)piperidine
1-(3-methoxyphenyl)-3-{[1-(oxan-4-yl)piperidin-3-yl]methyl}urea
5-(2-chloro-4-methoxyphenoxymethyl)-N-ethyl-N-(2-hydroxyethyl)-1H-pyrazole-3-carboxamide
2-{[(4-fluorophenyl)methyl](methyl)amino}-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
1-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]azetidin-3-yl}piperidine
7-(cyclopropylmethyl)-2-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}-2,7-diazaspiro[4.5]decane
N-{3-[2-(2-butyl-4-methyl-3-oxopiperazin-1-yl)-2-oxoethoxy]phenyl}propanamide
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(quinolin-4-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-{2-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
5-(1H-imidazol-2-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
2-(1-ethyl-1H-pyrazol-4-yl)-7-methyl-4-(3-methylpiperidine-1-carbonyl)quinoline
{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}urea
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethan-1-one
2-{2-[({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
(3R,4S)-4-[4-(2,3-dimethylquinoxaline-6-carbonyl)-1,4-diazepan-1-yl]oxolan-3-ol
1-(2,4-difluoro-3-methoxybenzoyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)(pyridin-4-ylmethyl)amine
6-(2-chloro-6-methoxyphenyl)-N,N-dimethylpyridine-3-carboxamide
1-(4-ethoxy-2-fluorophenyl)-3-(5-oxo-1-propylpyrrolidin-3-yl)urea
(3aS,6aS)-2-methyl-5-[3-(methylcarbamoyl)benzenesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholin-4-yl)-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-phenyl-N-(1-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(5-acetylthiophene-2-carbonyl)-4-benzyl-1,4-diazepan-5-one
1-{1-[(2-chloro-4,5-dimethoxyphenyl)methyl]piperidin-4-yl}piperidin-3-ol
2-[(3S,4R)-3-(propan-2-yl)-4-(propane-1-sulfonamido)pyrrolidin-1-yl]pyridine-3-carboxamide
[(4-methanesulfonylphenyl)methyl][(2-methoxyphenyl)methyl](prop-2-en-1-yl)amine
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-2-(4-propanoylphenoxy)acetamide
N-(2,2-difluoroethyl)-2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
1-cyclohexyl-4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazole
2-({[(3R,4R)-1-(2,6-difluoro-4-methoxybenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-methyl-8-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,5R)-3-methanesulfonyl-6-(2-methoxypyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-3-(methanesulfonylmethyl)piperidine
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[2-(morpholin-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-[3-chloro-2-(propan-2-yloxy)phenyl]-1-(oxan-4-yl)urea
2-(5-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
3,4,7-trimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide