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N-{3-oxo-3-[2-oxo-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propyl}acetamide
2-(4-methylphenyl)-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
N4-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-hydroxyethyl)-3-[5-(quinolin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[2-(1H-indol-3-yl)ethyl]propanamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(2,4-difluorophenyl)propan-1-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(quinoline-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
4-(1H-imidazol-1-ylmethyl)-5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazole
(1R,5R)-3-cyclobutanecarbonyl-6-(1H-imidazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-4-amino-N,N-diethyl-1-[(2E)-3-phenylprop-2-enoyl]pyrrolidine-2-carboxamide
2-[4-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
2-amino-N-[(3-ethoxyphenyl)methyl]-N-ethyl-4-phenylpyrimidine-5-carboxamide
3-amino-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-methylpropanamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2,8-dimethyl-4-[3-(piperidin-1-yl)azetidine-1-carbonyl]quinoline
(1S,5R)-6-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-{2,7-diazaspiro[4.5]decan-7-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrrolidine-1-sulfonamide
2-[(3aS,6aS)-1-(3-phenylpropyl)-octahydropyrrolo[3,4-b]pyrrol-5-yl]pyrimidin-4-amine
(2S,4R)-1-(2,2-diphenylethyl)-N-methyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
8-[2-(1-propylpiperidin-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N3-cyclooctyl-1-(2-methoxyethyl)-4-oxo-N5-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3,5-dicarboxamide
3-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}piperidin-2-one
N-[1-(3-methoxyphenyl)ethyl]-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
2-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1H-1,3-benzodiazole-4-carboxamide
2-(6-methoxypyridin-3-yl)-N-(propan-2-yl)benzamide
3-(3-methoxyphenyl)-N-[2-(propane-2-sulfonyl)ethyl]-1H-pyrazole-4-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]pyrrolidin-3-yl]methanol
3-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}-4H-chromen-4-one
1-cyclopentyl-4-oxo-N3-(propan-2-yl)-N5-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2-methyl-1H-indol-3-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1-propanoylpiperidine-3-carboxamide
1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
5-[(2S)-1-[5-(2-chlorophenyl)furan-2-carbonyl]pyrrolidin-2-yl]-3-ethyl-1,2,4-oxadiazole
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-methylpentane-1,2-dione
2-{2-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
(4aS,8aR)-6-(2,4-difluoro-3-methoxybenzoyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-cyclopropyl-1-(2-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
4-({4-[2-methyl-5-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
1-[(6-ethoxypyridin-3-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
5-chloro-3-methyl-N-{[4-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
5-methoxy-9-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecane
3-methyl-5-[(E)-2-phenylethenyl]pyridin-2-amine
7-(cyclobutylmethyl)-2-(quinolin-8-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[4-(pyridin-2-yl)butyl]acetamide