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4-[5-(3-methoxyphenoxymethyl)-3-methyl-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
8-{[4-(carboxymethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(3-fluorophenyl)-3-(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
(2S,4S)-4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-amido}-N-ethyl-1-(oxan-4-yl)pyrrolidine-2-carboxamide
ethyl 3-{[2-(3-methoxyphenyl)-1,3-benzoxazol-6-yl]formamido}propanoate
2-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
4-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)sulfonyl]benzonitrile
N-phenyl-5-[3-(pyridin-4-yl)azetidine-1-carbonyl]pyrimidin-2-amine
1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-ol
methyl 3-{2-[3-(morpholin-4-yl)-3-oxopropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propanoate
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(1-phenylcyclopropyl)piperidine-3-carboxamide
1-[(1R,2R)-2-(benzyloxy)cyclohexyl]-3-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
(2S)-2-[2-(2,4-difluorophenoxy)acetamido]-2-(2,3-difluorophenyl)acetic acid
N-(1-benzothiophen-2-ylmethyl)-1-{4-[(dimethylsulfamoyl)amino]phenyl}piperidin-4-amine
2-[4-chloro-2-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]acetic acid
N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
2-{4-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-1-benzylpiperazin-2-yl}ethan-1-ol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
N-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]-1-azabicyclo[2.2.2]octan-3-amine
2-(cyclohex-1-en-1-yl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
7-fluoro-2-methyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]quinoline-4-carboxamide
2-({4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)benzonitrile
7-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-1-oxa-7-azaspiro[3.5]nonane
7-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
1-(cyclopropylmethyl)-3-hydroxy-3-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}piperidin-2-one
3-(4-methylphenyl)-N-[2-(2-methylpropanesulfonyl)ethyl]-1H-pyrazole-5-carboxamide
3-(piperidin-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
2-oxo-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)pentanamide
4-(1H-imidazol-1-yl)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
8-(1-methyl-1H-pyrazole-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-[3-(oxolan-2-yl)propyl]piperidin-4-amine
methyl 2-[5-(6-hydroxy-2,6-dimethylheptyl)-4-phenyl-1H-imidazol-1-yl]acetate
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1,2,5-thiadiazole-3-carboxamide
2-benzyl-N-methyl-N-[4-(morpholin-4-yl)butyl]-1,3-benzoxazole-5-carboxamide
N,N-dimethyl-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine-1-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-oxo-4-phenylbutanamide
N-{[1-(furan-3-carbonyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
3,3-dimethyl-1-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]urea
N-(1-{7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-[(5-methylthiophen-2-yl)sulfonyl]pyrrolidine-2-carboxamide
5-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)pyrimidin-4-ol
3-(1H-indol-3-yl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}propan-1-one
N-methyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-(2-phenylethyl)acetamide
1-[5-(3,4-dimethylbenzoyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
1-(2-methylpropyl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-amine
2-benzyl-8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(4-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine