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(3S,9aR)-8-(3-chlorobenzoyl)-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}benzamide
1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-4-(3-chlorophenyl)piperazine
N-[1-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
4-[1-(2,4-difluorophenyl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-1-methylimidazolidin-2-one
2-{1-[(2-ethoxyphenyl)methyl]-4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
5-methyl-1-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[(1-benzyl-1H-pyrazol-4-yl)methyl]amino}propan-1-ol
3-fluoro-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-{2-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}methanesulfonamide
4-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-6-methylpyrimidin-2-amine
7-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-5-methylpyrazolo[1,5-a]pyrimidine
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}[(5-methylfuran-2-yl)methyl]amine
ethyl[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)sulfamoyl]methylamine
(3aR,6aR)-N-(1-acetylpiperidin-4-yl)-2-benzyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-4-(2-phenylethyl)piperazin-2-one
3-[1-(thiophene-3-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
3-[2-(dimethylamino)-2-(2-methylphenyl)acetamido]propanoic acid
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(pyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
3-(2-carboxyphenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
6-[(3S)-1-benzylpyrrolidin-3-yl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]azocane
2-methoxy-1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}ethan-1-one
5-benzyl-5-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-5-methyl-1,3-oxazole-4-carboxamide
1-(5-{[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
6-ethyl-N,1-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[2-(piperazin-1-yl)ethyl]-N-[1-(1,3-thiazol-5-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
5-methyl-6-(4-methylpiperazine-1-carbonyl)-N-[1-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
4-(hydroxymethyl)-1-(isoquinoline-5-carbonyl)piperidin-4-ol
ethyl 1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
(4aS,7aR)-N-benzyl-4-(furan-2-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(3aR,6aR)-2-cyclohexyl-5-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
N-(1H-indazol-4-yl)-4-(2-methylphenyl)-1,4-diazepane-1-carboxamide
2-[2-(1H-imidazol-1-yl)ethyl]-1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidine
1-{1-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(2-methyl-1,3-thiazol-4-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}acetamide
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one
N-[1-(hydroxymethyl)cyclopentyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(4aR,7aS)-4-{[5-(methylcarbamoyl)furan-2-yl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
8-{6-azaspiro[2.5]octane-1-carbonyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-3-(thiophen-2-yl)-1,2,4-oxadiazole
7-(2-methoxyethyl)-2-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one