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8-(6-methylpyridin-2-yl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,8-diazaspiro[4.5]decane
2-(6-chloro-8-methyl-4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
(3S,4S)-4-(naphthalen-2-yl)-1-(pyridin-2-ylmethyl)piperidin-3-ol
methyl 4-[(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazol-3-yl)formamido]butanoate
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl][1-(2-fluorophenyl)propan-2-yl]amine
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
ethyl 4-[(2-chlorophenyl)methyl]-1-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}piperidine-4-carboxylate
8-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-N,N-bis(propan-2-yl)benzamide
2-{5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
methyl 3-{[(2,3-dimethyl-1H-indol-5-yl)formamido]methyl}-5-[2-(1,3-thiazol-4-yl)acetamido]benzoate
2-(1-cyclopentyl-4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
3-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-3,9-diazaspiro[5.6]dodecan-10-one
2-{[2-(2-phenylethyl)morpholin-4-yl]methyl}-1H-1,3-benzodiazole
N-(2-methyl-3-{[1-(thiophen-2-yl)ethyl]carbamoyl}phenyl)furan-2-carboxamide
3-(4-chlorobenzoyl)-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
3-(4-cyano-2-fluorophenyl)-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
7-(cyclopropylmethyl)-2-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3R,4S)-4-cyclopropyl-1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]-1-(methoxymethyl)cyclopropane-1-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-{4-[6-(piperazin-1-yl)pyridin-2-yl]-1H-pyrazol-1-yl}acetamide
1-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)-3,5-dimethyl-1H-pyrazole
ethyl 2-[4-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)morpholin-3-yl]acetate
(2S)-4-methyl-2-{[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]formamido}pentanamide
4-fluoro-1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-4-ethoxypyrimidin-2-amine
N-[(1S,3R)-3-aminocyclopentyl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
(1S,5R)-3-(oxan-4-yl)-6-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-[2-(oxan-2-yl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
5-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
2-methoxy-N-(1-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(1-methyl-3-phenyl-1H-pyrazol-5-yl)urea
(1S,5R)-3-[4-(1H-imidazol-1-yl)butanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
4-(1H-imidazol-1-yl)-1-[2-(2-methylphenoxy)acetyl]piperidine-4-carboxylic acid
3-(oxolan-3-yl)-5-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazole
N-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-cyclobutanecarbonyl-1'-cyclohexyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-benzenesulfonamido-1-ethyl-2-methyl-N-[2-(pyrazin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(1,3-thiazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-(3-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}phenyl)morpholine
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
4-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-2-phenylpiperazine
(4aS,7aR)-1-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[(butan-2-yl)(cyclopentyl)amino]methyl}-6-methylpyridin-3-ol
4-(4-fluorophenyl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-4-ol
1-[2-(4-chlorophenyl)ethyl]-N-[2-(5-methylfuran-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl](2-methylprop-2-en-1-yl)amine
4-(morpholin-4-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pentanamide
(3aS,6aS)-2-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3aS,6aS)-2-[(3-phenoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid