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5-(1-cyclopropanecarbonylpyrrolidin-2-yl)-N-(1,3-dihydro-2-benzofuran-5-yl)thiophene-2-carboxamide
3-[5-(2-propoxyphenyl)-1,2,4-oxadiazol-3-yl]pyridazine
N,6-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
N-[4-(3-fluorophenyl)phenyl]-1-(1H-pyrazole-4-carbonyl)piperidine-3-carboxamide
2-(3-methoxypropyl)-9-(3-phenylpropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
8-(3-methyl-1-benzothiophene-2-carbonyl)-1-oxa-8-azaspiro[4.5]decane
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-(methylamino)pyridine-4-carboxamide
1-(2-methoxy-6-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
3-{5-[(2R)-2-amino-3-methoxypropanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-ethyl-7-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.4]nonane
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](1,4-dioxan-2-ylmethyl)methylamine
N-cyclopentyl-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
4-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-[2-(3-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
propan-2-yl 4-chloro-3-[2-(4-chloro-1H-pyrazol-1-yl)acetamido]benzoate
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-5-methyl-1,3-oxazole-4-carboxamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(3-hydroxyquinoxalin-2-yl)propanamide
4-methyl-1-{3'-oxo-4'-propyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pentane-1,2-dione
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(1-{[1-(2-ethylhexyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[(3-methylthiophen-2-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-(1-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
1-(pyrimidin-5-yl)-1H-1,3-benzodiazole
3-({5-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}methyl)pyridine
2-(5-acetylthiophen-3-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
9-(2-propoxypropanoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-2,6-dimethylpyridine-4-carboxamide
2-(4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
2,3-dimethyl-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-1H-indole-5-carboxamide
({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]amine
1-(2-methylpropyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]piperidin-4-amine
3-(piperidin-1-ylmethyl)-1-(quinolin-5-ylmethyl)pyrrolidin-3-ol
3-[(3R,4S)-1-(2-fluoro-6-methoxybenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-ethyl-3-methyl-4-[4-(1H-pyrazol-4-yl)butanoyl]piperazin-2-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-hydroxy-2-methylbenzamide
3-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
ethyl 1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylfuran-2-carboxamide
1-[(2-methylpyrimidin-5-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
methyl 3-(cyclobutylmethoxy)-5-{[(1r,4r)-4-hydroxycyclohexyl]carbamoyl}benzoate
4-(2,6-dimethylpyridin-3-yl)-2-[4-(prop-2-en-1-yl)piperazin-1-yl]pyrimidine
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-8-methyl-2-(1H-pyrazol-4-yl)quinoline
7-(3-fluoropyridin-4-yl)-2-methyl-N-(oxan-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 1-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-(3-methylbutyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
2-amino-4-[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-5H,6H,7H,8H,9H-cyclohepta[b]pyridine-3-carbonitrile
3-chloro-5-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[4-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]-1-(pyrrolidin-1-yl)ethan-1-one
1-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-2-one